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Cat. No. Product Name Target Signaling Pathways
T12398 MP7

PDK1 抑制剂,PDK1 inhibitor

PDK PI3K/Akt/mTOR signaling
MP7 (PDK1 inhibitor) 是磷酸肌醇依赖性激酶-1 (PDK1) 抑制剂。
T11872L LMP744 hydrochloride

NSC706744 hydrochloride,MJ-III65 hydrochloride

Topoisomerase DNA Damage/DNA Repair
LMP744 hydrochloride (NSC-706744 hydrochloride) 是一种是拓扑异构酶 1 抑制剂,显示出抗肿瘤的活性。
T13172 TMP780

ROR Metabolism
TMP780 is an inverse RORγt agonist (IC50: 13 nM). RORγt is a tractable drug target for the treatment of cutaneous inflammatory disorders.
T11872 LMP744

NSC706744,MJ-III65

Others Others
LMP744 is a DNA intercalator and Topoisomerase I (Top1) inhibitor with antitumor activity.
T13172L TMP778

Others Others
TMP778 is an effective and selective RORγt inverse agonist (IC50: 7 nM in FRET assay).
T81921 LMP7-IN-2

LMP7-IN-2, 作为LMP7抑制剂,适用于相关炎症性疾病与失调的治疗。

化合物

MP7
Cat.No: T12398
Synonym: PDK1 抑制剂,PDK1 inhibitor
Target: PDK
LMP744 hydrochloride
Cat.No: T11872L
Synonym: NSC706744 hydrochloride,MJ-III65 hydrochloride
Target: Topoisomerase
TMP780
Cat.No: T13172
Synonym:
Target: ROR
LMP744
Cat.No: T11872
Synonym: NSC706744,MJ-III65
Target: Others
TMP778
Cat.No: T13172L
Synonym:
Target: Others
LMP7-IN-2
Cat.No: T81921
Synonym:
Target:
TargetMol Loading
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