Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T12028 | MGAT2-IN-1 | Others | Others |
MGAT2-IN-1 is an orally active monoacylglycerol acyltransferase (MGAT2)inhibitor (human and mouse MGAT2 with IC50 of 7.8 and 2.4 nM , respectively). | |||
T81802 |
MGAT2-IN-4
|
||
MGAT2-IN-4(compound 33)是一种针对单酰基甘油转移酶2(MGAT2)的抑制剂,显示出良好的肝脏代谢稳定性,适用于肥胖症、糖尿病以及非酒精性脂肪性肝炎(NASH)的研究。 | |||
T82848 |
BMS-986172
|
Acyltransferase | Metabolism |
BMS-986172是一种高选择性的口服MGAT2抑制剂,针对hMGAT2和mMGAT2显示出的IC50分别为4.6 nM和20 nM。该化合物在体外具有较长的半衰期(T1/2>120分钟),能够减少食物摄入和体重。BMS-986172在治疗肥胖和NASH等代谢性疾病方面显示出研究潜力。 |