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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T7460 α-Cyano-4-hydroxycinnamic acid

α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基

Monocarboxylate transporter Membrane transporter/Ion channel
α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) 是非竞争性单羧酸盐转运蛋白 (MCTs) 抑制剂,可抑制线粒体丙酮酸转运蛋白,Ki 值为 6.3 μM。它可作为基质辅助激光解吸电离-飞行时间质谱 (MALDI-TOF) 分析的基质,可以促进肽离子化。
T39767 AR-C141990 hydrochloride

AR-C141990 hydrochloride

AR-C141990 hydrochloride is a potent inhibitor of lactate transporters known as monocarboxylate transporters (MCTs). It has pK i values of 7.6 and 6.6 for MCT-1 and MCT-2, respectively. Additionally, this compound exhibits immunosuppressive properties and effectively inhibits the graft versus host response.

化合物

α-Cyano-4-hydroxycinnamic acid
Cat.No: T7460
Synonym: α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基
Target: Monocarboxylate transporter
AR-C141990 hydrochloride
Cat.No: T39767
Synonym: AR-C141990 hydrochloride
Target:
Cat. No. Product Name Target Signaling Pathways
TN2252 Syrosingopine

Dopamine Receptor GPCR/G Protein; Neuroscience
Syrosingopine 是 MCT1和 MCT4双重抑制剂,对 MCT4 的效力高 60 倍,可防止乳酸和 H+ 流出。它是可口服抗高血压药物,联合二甲双胍具有研究癌症疾病的潜力。

天然产物

Syrosingopine
Cat.No: TN2252
Synonym:
Target: Dopamine Receptor
TargetMol Loading
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