首页 工具
登录
购物车

搜索结果

Search Results for " mch-1 antagonist 1 "

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T11964 MCH-1 antagonist 1

P450 Metabolism
MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).
T8004 SNAP 94847 hydrochloride

GPR; Melanin-concentrating Hormone Receptor (MCHR) Endocrinology/Hormones; GPCR/G Protein
SNAP 94847 hydrochloride 是一种选择性黑色素浓缩激素受体1 拮抗剂,Ki 为 2.2 nM,具有抗抑郁样活性。它是 MCH 诱发的肌醇磷酸形成的高亲和力拮抗剂 ,pA2为 7.81
T15450 GW-803430

GW-3430

Others Others
GW-803430 is a potent and selective antagonist of melanin-concentrating hormone receptor 1 (MCH R1) (pIC50: 9.3). GW-803430 is orally active in an animal model of obesity.
T7749 ALB-127158

ALB-127158(a) 是一种有效的选择性黑色素浓缩激素 1 (MCH1) 受体拮抗剂,可能是炎症性肠病 (IBD) 的潜在治疗方法

化合物

MCH-1 antagonist 1
Cat.No: T11964
Synonym:
Target: P450
SNAP 94847 hydrochloride
Cat.No: T8004
Synonym:
Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)
GW-803430
Cat.No: T15450
Synonym: GW-3430
Target: Others
ALB-127158
Cat.No: T7749
Synonym:
Target:
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼