Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1735 |
Lurasidone hydrochloride
Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496 |
Dopamine Receptor; 5-HT Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Lurasidone hydrochloride (Lurasidone HCl) 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM,用于治疗精神分裂症和双相情感障碍。它也是5-HT1A 受体的部分激动剂,IC50值为 6.75 nM。 | |||
T11893L |
Lurasidone metabolite 14326 hydrochloride
Lurasidone metabolite 14326 hydrochloride (186204-33-1 free base) |
Others | Others |
Lurasidone metabolite 14326 hydrochloride, an active metabolite of the atypical antipsychotic Lurasidone, maintains its significant function in pharmacological efficacy. | |||
T11892 |
Lurasidone D8 Hydrochloride
SM-13496 D8 |
Others | Others |
Lurasidone D8 Hydrochloride is an inhibitor of Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C, and is the deuterium labeled Lurasidone. | |||
T13760 |
Lurasidone Metabolite 14283 hydrochloride
|
Others | Others |
Lurasidone Metabolite 14283 hydrochloride is a major active metabolite of Lurasidone. | |||
TMIH-0315 |
Lurasidone Inactive Metabolite 14283-d8
5α/6α-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers) |
||
Lurasidone Inactive Metabolite 14283-d8 是 Lurasidone Inactive Metabolite 14283 的氘代化合物。Lurasidone Inactive Metabolite 14283 的 CAS 号为 186204-31-9。 | |||
TMIH-0316 |
Lurasidone Inactive Metabolite 14326-d8
5β/6β-Hydroxy Lurasidone-d8 Hydrochloride (Mixture of Diastereomers) |
||
Lurasidone Inactive Metabolite 14326-d8 是 Lurasidone Inactive Metabolite 14326 的氘代化合物。Lurasidone Inactive Metabolite 14326 的 CAS 号为 186204-33-1。 | |||
TMIH-0314 |
Lurasidone-d8 HCl
|
||
Lurasidone-d8 HCl 是 Lurasidone HCl 的氘代化合物。Lurasidone HCl 的 CAS 号为 367514-88-3。Lurasidone hydrochloride 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM,用于治疗精神分裂症和双相情感障碍。它也是5-HT1A受体的部分激动剂,IC50值为 6.75 nM。 |