Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T25672 |
Lesopitron
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Lesopitron 是一种具有突触前和突触后5-HT1A 激动剂活性的抗焦虑剂,在大鼠社会交往和狨猴焦虑模型中比5-HT1A 激动剂更有效。Lesopitron 能对抗苯二氮卓类药物戒断引起的啮齿动物的焦虑且急性毒性很低,不会增强酒精或巴比妥类药物的作用。 | |||
T11839L |
Lesopitron HCl
Lesopitron HCl(132449-89-9 Free base) |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Lesopitron HCl 是一种5-HT1A 受体激动剂,具有抗焦虑化作用,可逆转与小鼠可卡因戒断相关的黑暗回避行为。 | |||
T11839 |
Lesopitron dihydrochloride
E4424 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist. |