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Cat. No. Product Name Target Signaling Pathways
T6047 Ralimetinib dimesylate

LY2228820 dimesylate,Ralimetinib,LY2228820,Ralimetinib Mesylate

Apoptosis; p38 MAPK; Autophagy Apoptosis; Autophagy; MAPK
Ralimetinib dimesylate (LY2228820 dimesylate) 是一种选择性,ATP 竞争性的 p38 MAPK α/β抑制剂,IC50分别为5.3 和 3.2 nM。
T16721 Ralimetinib

LY2228820

Others Others
Ralimetinib selectively inhibits phosphorylation of MK2 (Thr334) and has no effect on phosphorylation of p38α MAPK, JNK, ERK1/2, c-Jun, ATF2, or c-Myc. Ralimetinib is an effective and selective, ATP-competitive inhibitor of p38 MAPK α/β (IC50s: 5.3 and 3.

化合物

Ralimetinib dimesylate
Cat.No: T6047
Synonym: LY2228820 dimesylate,Ralimetinib,LY2228820,Ralimetinib Mesylate
Target: Apoptosis, p38 MAPK, Autophagy
Ralimetinib
Cat.No: T16721
Synonym: LY2228820
Target: Others
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