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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16348 |
NS5806
NS-5806 |
Potassium Channel | Membrane transporter/Ion channel |
NS5806 是钾电流的激活剂,可增加 KV4.3/KChIP2峰值电流幅度,EC50值为 5.3 μM。它会在包含 KChIP2 的通道复合体中降低 KV4.2 和 KV4.3 电流衰减。 | |||
T80500 |
Jingzhaotoxin-X
JZTX-X |
Potassium Channel | Membrane transporter/Ion channel |
Jingzhaotoxin-X (JZTX-X) is a selective inhibitor of Kv4.2 and Kv4.3 potassium channels, inducing persistent mechanical hyperalgesia. | |||
T80054 |
Phrixotoxin 2
|
Potassium Channel | Membrane transporter/Ion channel |
Phrixotoxin 2为具有高选择性的KV4.2与KV4.3通道阻断剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4550 |
Ajmaline
Cardiorythmine,Raugalline,阿义吗啉,阿义马林,Tachmalin,(+)-Ajmaline |
Sodium Channel | Membrane transporter/Ion channel |
Ajmaline (Cardiorythmine) 是一种钠通道阻断剂,属于1A 类抗心律失常剂。Ajmaline 阻断 HERG 电流,在 HEK 细胞的 IC50为 1 μM,爪蟾卵母细胞的IC50为 42.3 μM。Ajmaline 在室性心动过速方面具有研究价值。 |