Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3015 |
Olaparib
AZD2281,奥拉帕尼,KU0059436 |
Mitophagy; PARP; Autophagy | Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair |
Olaparib (KU0059436) 是 PARP1/PARP2 的小分子抑制剂 (IC50=5/1 nM),对 PARP tankyrase-1 的抑制活性较弱 (IC50=1.5 μM),具有选择性和口服活性。Olaparib 具有自噬和线粒体自噬激活活性。 | |||
T12292 |
Olaparib-d5
KU0059436 D5,AZD2281 D5,Olaparib D5 |
Others | Others |
Olaparib D5 is a deuterium labeled Olaparib. Olaparib is a potent and oral inhibitor of PARP. |