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抑制剂 & 化合物

9

天然产物

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Cat. No. Product Name Target Signaling Pathways
T11783 KSI-3716

c-Myc Cell Cycle/Checkpoint
KSI-3716 is an inhibitor of c-Myc.
T71011 Perfluorinated SAHA

Perfluorinated SAHA is an HDAC inhibitor for use in cancer treatment regimens, with demonstrated greater antiproliferative properties than SAHA . PFSAHA has also been shown to have higher selectivity for PA3774, an HDAC-like enzyme from P. aeruginosa, as well as other HDACs, which may prove beneficial for developing novel chemotherapeutic treatments for cancer.
T82929 AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG

AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG 促进骨化作用。该化合物适用于研究成骨缺陷或骨矿物质密度(BMD)降低相关疾病,如骨质疏松症。
T35579 PKSI-527

PKSI-527 is an inhibitor of plasma kallikrein (Ki = 0.81 μM). It is selective for plasma kallikrein over glandular kallikrein, plasmin, thrombin, urokinase, and Factor Xa (Kis = >500, 390, >500, 200, and >500 μM, respectively). PKSI-527 reduces bradykinin generation induced by kaolin and λ-carrageenan ex vivo in human plasma. It also prolongs partial thromboplastin and euglobulin clot lysis times. In vivo, PKSI-527 (300 mg/kg per day) reduces hyperplasia, pannus formation, and infiltration of in...

化合物

KSI-3716
Cat.No: T11783
Synonym:
Target: c-Myc
Perfluorinated SAHA
Cat.No: T71011
Synonym:
Target:
AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG
Cat.No: T82929
Synonym:
Target:
PKSI-527
Cat.No: T35579
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2967 Pinobanksin 3-acetate

3-O-Acetylpinobanksin

Others; Antioxidant Others; oxidation-reduction
Pinobanksin 3-acetate (3-O-Acetylpinobanksin) 是一种短叶松素酯衍生物,是一种强抗氧化剂,存在于向日葵和蜂蜜中,可以抑制低密度脂蛋白的过氧化.
TN3860 Dihydroperaksine

Others Others
Dihydroperaksine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN3860,CAS号为 16100-84-8。Dihydroperaksine可用作对照参考。
TN4789 Pinobanksin 3-O-propanoate

Others Others
Pinobanksin 3-O-propanoate is a natiral product from forest trees.
TN2910 3,7-O-Diacetylpinobanksin

Others Others
3,7-O-Diacetylpinobanksin是一种天然产物,属于松科松属,其产品编号为 TN2910,CAS号为 103553-98-6。3,7-O-Diacetylpinobanksin可用作对照参考。
TN4790 Pinobanksin 5-methyl ether

Others Others
Pinobanksin 5-methyl ether can induce detoxification genes.
TN2076 Pinobanksin

短叶松素

Others Others
Pinobanksin and some of its ester derivatives from Sonoran propolis have apoptotic induction in a B-cell lymphoma cell line.
TN6030 Peraksine

Peraksine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN6030,CAS号为 15527-80-7。Peraksine可用作对照参考。
TN2568 10-Hydroxydihydroperaksine

Others Others
10-Hydroxydihydroperaksine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN2568,CAS号为 451478-47-0。10-Hydroxydihydroperaksine可用作对照参考。
TN5486 Pinobanksin 3-(2-methyl)butyrate

Apoptosis Apoptosis
Pinobanksin 3-(2-methyl)butyrate 是 Pinobanksin 衍生物。pinobanksin 是一种细胞凋亡诱导剂,可诱导 F6细胞凋亡。

天然产物

Pinobanksin 3-acetate
Cat.No: TN2967
Synonym: 3-O-Acetylpinobanksin
Target: Others, Antioxidant
Dihydroperaksine
Cat.No: TN3860
Synonym:
Target: Others
Pinobanksin 3-O-propanoate
Cat.No: TN4789
Synonym:
Target: Others
3,7-O-Diacetylpinobanksin
Cat.No: TN2910
Synonym:
Target: Others
Pinobanksin 5-methyl ether
Cat.No: TN4790
Synonym:
Target: Others
Pinobanksin
Cat.No: TN2076
Synonym: 短叶松素
Target: Others
Peraksine
Cat.No: TN6030
Synonym:
Target:
10-Hydroxydihydroperaksine
Cat.No: TN2568
Synonym:
Target: Others
Pinobanksin 3-(2-methyl)butyrate
Cat.No: TN5486
Synonym:
Target: Apoptosis
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