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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11783 | KSI-3716 | c-Myc | Cell Cycle/Checkpoint |
KSI-3716 is an inhibitor of c-Myc. | |||
T71011 | Perfluorinated SAHA | ||
Perfluorinated SAHA is an HDAC inhibitor for use in cancer treatment regimens, with demonstrated greater antiproliferative properties than SAHA . PFSAHA has also been shown to have higher selectivity for PA3774, an HDAC-like enzyme from P. aeruginosa, as well as other HDACs, which may prove beneficial for developing novel chemotherapeutic treatments for cancer. | |||
T82929 |
AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG
|
||
AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG 促进骨化作用。该化合物适用于研究成骨缺陷或骨矿物质密度(BMD)降低相关疾病,如骨质疏松症。 | |||
T35579 |
PKSI-527
|
||
PKSI-527 is an inhibitor of plasma kallikrein (Ki = 0.81 μM). It is selective for plasma kallikrein over glandular kallikrein, plasmin, thrombin, urokinase, and Factor Xa (Kis = >500, 390, >500, 200, and >500 μM, respectively). PKSI-527 reduces bradykinin generation induced by kaolin and λ-carrageenan ex vivo in human plasma. It also prolongs partial thromboplastin and euglobulin clot lysis times. In vivo, PKSI-527 (300 mg/kg per day) reduces hyperplasia, pannus formation, and infiltration of in... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN2967 |
Pinobanksin 3-acetate
3-O-Acetylpinobanksin |
Others; Antioxidant | Others; oxidation-reduction |
Pinobanksin 3-acetate (3-O-Acetylpinobanksin) 是一种短叶松素酯衍生物,是一种强抗氧化剂,存在于向日葵和蜂蜜中,可以抑制低密度脂蛋白的过氧化. | |||
TN3860 |
Dihydroperaksine
|
Others | Others |
Dihydroperaksine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN3860,CAS号为 16100-84-8。Dihydroperaksine可用作对照参考。 | |||
TN4789 |
Pinobanksin 3-O-propanoate
|
Others | Others |
Pinobanksin 3-O-propanoate is a natiral product from forest trees. | |||
TN2910 |
3,7-O-Diacetylpinobanksin
|
Others | Others |
3,7-O-Diacetylpinobanksin是一种天然产物,属于松科松属,其产品编号为 TN2910,CAS号为 103553-98-6。3,7-O-Diacetylpinobanksin可用作对照参考。 | |||
TN4790 |
Pinobanksin 5-methyl ether
|
Others | Others |
Pinobanksin 5-methyl ether can induce detoxification genes. | |||
TN2076 |
Pinobanksin
短叶松素 |
Others | Others |
Pinobanksin and some of its ester derivatives from Sonoran propolis have apoptotic induction in a B-cell lymphoma cell line. | |||
TN6030 |
Peraksine
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||
Peraksine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN6030,CAS号为 15527-80-7。Peraksine可用作对照参考。 | |||
TN2568 |
10-Hydroxydihydroperaksine
|
Others | Others |
10-Hydroxydihydroperaksine是一种天然产物,属于夹竹桃科萝芙木属,其产品编号为 TN2568,CAS号为 451478-47-0。10-Hydroxydihydroperaksine可用作对照参考。 | |||
TN5486 |
Pinobanksin 3-(2-methyl)butyrate
|
Apoptosis | Apoptosis |
Pinobanksin 3-(2-methyl)butyrate 是 Pinobanksin 衍生物。pinobanksin 是一种细胞凋亡诱导剂,可诱导 F6细胞凋亡。 |