购物车

搜索结果

Search Results for " itp "

6

抑制剂 & 化合物

1

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T40359 Thio-ITP

6-Thio-ITP,Thio-ITP,6-Mercaptopurine-riboside-5'-triphosphate,6-Thioinosine 5′-triphosphate

Thio-ITP, also known as 6-Thioinosine 5'-triphosphate, is a competitive inhibitor of RNA polymerase activity. It exhibits a strong apparent affinity towards the polymerases, with Ki values of 40.9 μM for RNA polymerase I and 38.0 μM for RNA polymerase II.
T70691 ITP-2

ITP-2 is a selective activator of hERG channels. ITP-2 causes large depolarizing shifts in the midpoint of voltage-dependent inactivation and hyperpolarizing shifts in the voltage-dependence of activation.
T70689 MEN-10354

MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.
T32088 Sovleplenib

HMPL 523,HMPL523,HMPL-523

Syk Angiogenesis; Tyrosine Kinase/Adaptors
Sovleplenib (HMPL523) 是一种可口服且具有选择性和高效性的脾酪氨酸激酶 SYK 抑制剂,IC50 为 25 nM。Sovleplenib 具有抗肿瘤活性,可用于免疫性血小板减少症(ITP)的研究。
T82893 Bevifimod

PRTX-100

Bevifimod (PRTX-100),一种高度纯化的葡萄球菌蛋白A (SpA),主要用于特发性血小板减少性紫癜(ITP)的研究。
T77084 Mezagitamab

Mezagitamab (TAK-079) 是一种 IgG1λ 类型的抗CD38单克隆抗体。其通过促进抗体和补体依赖性的细胞毒性,来耗尽表达CD38的肿瘤细胞,显示出在复发/难治性多发性骨髓瘤 (RRMM) 及原发性血小板减少性紫癜 (ITP) 等疾病中的治疗潜力。

化合物

Thio-ITP
Cat.No: T40359
Synonym: 6-Thio-ITP,Thio-ITP,6-Mercaptopurine-riboside-5'-triphosphate,6-Thioinosine 5′-triphosphate
Target:
ITP-2
Cat.No: T70691
Synonym:
Target:
MEN-10354
Cat.No: T70689
Synonym:
Target:
Sovleplenib
Cat.No: T32088
Synonym: HMPL 523,HMPL523,HMPL-523
Target: Syk
Bevifimod
Cat.No: T82893
Synonym: PRTX-100
Target:
Mezagitamab
Cat.No: T77084
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4897 Inosine-5'-triphosphate trisodium salt

ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt

Others; Endogenous Metabolite Metabolism; Others
Inosine-5'-triphosphate trisodium salt (ITP) 是三磷酸核苷,能够作为 ATPases 和 GTPases 的底物。

天然产物

Inosine-5'-triphosphate trisodium salt
Cat.No: T4897
Synonym: ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt
Target: Others, Endogenous Metabolite
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼