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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T11619 IDO-IN-5

NLG-1489

IDO Metabolism
IDO-IN-5 is an indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 1-10 μM).
T11901 IDO1-IN-5

IDO; Indoleamine 2,3-Dioxygenase (IDO) Metabolism
IDO1-IN-5 是可透过血脑屏障的、选择性的IDO1抑制剂,能够与缺乏血红素的 apo-IDO1 结合,但无法与成熟血红素的 IDO1 结合。
T12801 (S)-IDO1-IN-5

Others Others
(S)-IDO1-IN-5 is an active S-isomer of IDO1-IN-5. (S)-IDO1-IN-5 binds to IDOL(IC50 value less than 1.5 µΜ).
T12668 (Rac)-IDO1-IN-5

Others Others
(Rac)-IDO1-IN-5 is a racemate of IDO1-IN-5, a potent, selective, and brain-penetrating inhibitor of Indoleamine 2,3-Dioxygenase 1 (IDO1) activity. It specifically binds to apo-IDO1, which lacks heme, instead of mature heme-bound IDO1.
T62130 IDO-IN-16

IDO-IN-16 (compound 5) 是一种 IDO 抑制剂 (IC50: 36 nM)。

化合物

IDO-IN-5
Cat.No: T11619
Synonym: NLG-1489
Target: IDO
IDO1-IN-5
Cat.No: T11901
Synonym:
Target: IDO, Indoleamine 2,3-Dioxygenase (IDO)
(S)-IDO1-IN-5
Cat.No: T12801
Synonym:
Target: Others
(Rac)-IDO1-IN-5
Cat.No: T12668
Synonym:
Target: Others
IDO-IN-16
Cat.No: T62130
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5S0053 Coptisine

黄连碱,Coptisin

Indoleamine 2,3-Dioxygenase (IDO) Metabolism
Coptisine (Coptisin) 是一种从黄连中分离到的生物碱,是非竞争性的IDO 抑制剂,Ki=为 5.8 μM,IC50=6.3 μM。

天然产物

Coptisine
Cat.No: T5S0053
Synonym: 黄连碱,Coptisin
Target: Indoleamine 2,3-Dioxygenase (IDO)
TargetMol Loading
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