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Search Results for " hematoxylin "

3

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T2178 AMI5

AMI 5,Eosin Y Disodium,AMI-5

Others Others
AMI5 (Eosin Y Disodium) 是一种具有可溶性的酸性红色染料分子。它常用于机合成中的光氧化还原催化剂。
T15469 Hematein

Hydroxybrasilein

Wnt/beta-catenin; Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Stem Cells
Hematein 抑制Akt/PKB Ser129磷酸化,Wnt/TCF 途径,并增加癌症细胞的凋亡。Hematein 是苏木精的氧化产物,也是变构酪蛋白激酶II 抑制剂(IC50:0.74μM)。
T71082 DW532

DW532 is one of simplified analogues of hematoxylin that has shown broad-spectrum inhibition on tyrosine kinases and in vitro anti-cancer activities. DW532 inhibited EGFR and VEGFR2 in vitro kinase activity (the IC50 values were 4.9 and 5.5 μmol/L, respectively), and suppressed their downstream signaling. DW532 dose-dependently inhibited tubulin polymerization via direct binding to tubulin, thus disrupting the mitotic spindle assembly and leading to abnormal cell division. In a panel of human ca...

化合物

AMI5
Cat.No: T2178
Synonym: AMI 5,Eosin Y Disodium,AMI-5
Target: Others
Hematein
Cat.No: T15469
Synonym: Hydroxybrasilein
Target: Wnt/beta-catenin, Akt
DW532
Cat.No: T71082
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1686 Hematoxylin

苏木精,Hydroxybrazilin,Natural Black 1,Haematoxylin

Beta Amyloid; Others Neuroscience; Others
Hematoxylin (Natural Black 1) 是一种天然存在的类黄酮化合物,衍生自木柴树Haematoxylon campechianum。它是一种组织学上的核染色剂,也是一种有效的Aβ42原纤维形成的抑制剂,IC50=1.6 µM。

天然产物

Hematoxylin
Cat.No: T1686
Synonym: 苏木精,Hydroxybrazilin,Natural Black 1,Haematoxylin
Target: Beta Amyloid, Others
TargetMol Loading
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