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2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3504 |
AZD5153 6-Hydroxy-2-naphthoic acid
AZD5153,AZD5153结晶体(API形式),AZD-5153 HNT salt |
Epigenetic Reader Domain | Chromatin/Epigenetic |
AZD5153 6-Hydroxy-2-naphthoic acid (AZD5153) 是 AZD5153的6-羟基-2-萘甲酸盐形式。AZD5153是一种有口服活性的选择性 BET/BRD4溴结构域抑制剂,对BRD4的IC50值为1.7nM。 | |||
T65242 |
HNTU
|
||
O-(5-Norbornene-2,3-dicarboximido)-N,N,N',N'-tetramethyluronium Hexafluorophosphate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65242,CAS号为 208462-94-6。 | |||
T78954 |
hNTS1R agonist-1
|
Neurotensin Receptor | GPCR/G Protein |
hNTS1R agonist-1 (Compound 10)为能穿透血脑屏障的hNTS1R全激动剂(Ki:6.9 nM)。它能提升帕金森病(PD)模型小鼠的运动能力及记忆。作为一种Neurotensin(8-13)类似物,hNTS1R agonist-1同时具有神经保护作用。 |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-00357 |
HNT/NTM Protein, Human, Recombinant (His)
HNT,NTRI,IGLON2,neurotrimin |
Human | HEK293 Cells |
HNT/NTM Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 32.3 kDa and the accession number is Q9P121-3. | |||
TMPY-00355 |
HNT/NTM Protein, Human, Recombinant (hFc)
neurotrimin,NTRI,IGLON2,HNT |
Human | HEK293 Cells |
HNT/NTM Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 57.6 kDa and the accession number is Q9P121-1. |