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Cat. No. Product Name Target Signaling Pathways
T21867 BI-6015

2-甲基-1-(2-甲基-5-硝基苯基磺酰基)-1H-苯并[D]咪唑

Others Others
BI 6015 是肝细胞核因子 (HNF) 拮抗剂,可抑制已知 HNF 靶基因的表达。它利用 HNF 拮抗作用,降低胰岛素启动子活性,可用于研究癌症和糖尿病。
T15389L Glucagon (1-29), bovine, human, porcine hydrochloride

盐酸胰高血糖素,Porcine glucagon hydrochloride,Glucagon hydrochloride

Glucocorticoid Receptor; Glucagon Receptor Endocrinology/Hormones; GPCR/G Protein
Glucagon (1-29), bovine, human, porcine hydrochloride 是一种由胰腺 α 细胞产生的多肽激素。它可激活 HNF 并促进 HNF 磷酸化,促进糖异生。
T11131 DW14800

Histone Methyltransferase Chromatin/Epigenetic
DW14800是PRMT5的抑制剂(IC50 = 17 nM),能增强HNF的转录,并降低H4R3me2s 的水平。
T15389 Glucagon (1-29), bovine, human, porcine

胰高血糖素,Porcine glucagon,Glucagon

Others Others
Glucagon is a peptide hormone, produced by pancreatic α-cells. Glucagon reduces the activity of HNF-4. Glucagon stimulates gluconeogenesis. Glucagon enhances HNF phosphorylation.

化合物

BI-6015
Cat.No: T21867
Synonym: 2-甲基-1-(2-甲基-5-硝基苯基磺酰基)-1H-苯并[D]咪唑
Target: Others
Glucagon (1-29), bovine, human, porcine hydrochloride
Cat.No: T15389L
Synonym: 盐酸胰高血糖素,Porcine glucagon hydrochloride,Glucagon hydrochloride
Target: Glucocorticoid Receptor, Glucagon Receptor
DW14800
Cat.No: T11131
Synonym:
Target: Histone Methyltransferase
Glucagon (1-29), bovine, human, porcine
Cat.No: T15389
Synonym: 胰高血糖素,Porcine glucagon,Glucagon
Target: Others
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