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Cat. No. Product Name Target Signaling Pathways
T10603 BRD-6929

HIV Protease; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
BRD-6929 是一种选择性的脑渗透性的HDAC1和HDAC2抑制剂 ,IC50值为 1 和 8 nM。它对 HDAC1 和 HDAC2 有高亲和力,Ki 值为  0.2 和 1.5 nM。它可研究情绪相关行为。
T5347 CXD101

CXD-101

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
CXD101 是一种选择性和具有口服活性的 I 类HDAC 抑制剂,有抗肿瘤活性,对HDAC1、HDAC2和HDAC3的IC50分别为 63、570 和 550 nM。
T26355 ZYJ-34c

ZYJ 34c,ZYJ34c

ZYJ-34c is a potent oral antitumor activities histone deacetylase inhibitor (HDACi).
T71917 FFK29

FFK29 is a synthetic class II HDACi (Histone deacetylase inhibitors) which have have recently emerged as novel therapeutic options for treating various protozoan and parasitic diseases. While these HDACi demonstrated a negligible effect on the viability of mature cysts, Acanthamoeba encystation was significantly inhibited by these HDACi. In conclusion, these synthetic HDACi demonstrated potent amoebicidal effects and inhibited the growth and encystation of Acanthamoeba, thus highlighting their e...
T26354 ZYJ-25e

ZYJ 25e

ZYJ-25e is an oral histone deacetylase inhibitor (HDACi) with potent antitumor activities.
T26356 ZYJ-34v

ZYJ-34v is an oral histone deacetylase inhibitor (HDACi) with potent antitumor activities.
T62041 XP5

XP5 是一种有效的、具有口服活性的HDAC6抑制剂(IC50= 31 nM)。XP5高效抑制各种癌细胞系(包括抗 HDACi 的 YCC3/7 胃癌细胞)的增殖 (IC50=0.16-2.31 μM)。
T70190 Tinostamustine HCl

Tinostamustine, also known as EDO-S101, is an alkylatlng histone-deacetylase inhibitor (HDACi) fusion molecule. EDO-S101 is a functional pan-histone-deacetylase inhibitor and is assumed to potentiate the alkylating activity of the compound and/or may help to overcome resistance to other therapeutic agents.
T61209 HDAC-IN-27

HDAC-IN-27 是一种有效的口服活性HDACI 类选择性抑制剂,对 HDAC1-3 的 IC50值范围为 0.43 至 3.01 nM。抗急性髓系白血病 (AML) 活性。

化合物

BRD-6929
Cat.No: T10603
Synonym:
Target: HIV Protease, HDAC
CXD101
Cat.No: T5347
Synonym: CXD-101
Target: HDAC
ZYJ-34c
Cat.No: T26355
Synonym: ZYJ 34c,ZYJ34c
Target:
FFK29
Cat.No: T71917
Synonym:
Target:
ZYJ-25e
Cat.No: T26354
Synonym: ZYJ 25e
Target:
ZYJ-34v
Cat.No: T26356
Synonym:
Target:
XP5
Cat.No: T62041
Synonym:
Target:
Tinostamustine HCl
Cat.No: T70190
Synonym:
Target:
HDAC-IN-27
Cat.No: T61209
Synonym:
Target:
TargetMol Loading
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