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Cat. No. | Product Name | Target | Signaling Pathways |
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T74013 |
Geldanamycin-FITC
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Geldanamycin-FITC 是一种格尔达霉素荧光探针,可用于HSP90抑制剂的荧光偏振分析。Geldanamycin-FITC 也可用于细胞表面HSP90的检测。储存方式:避光。 | |||
T37377 | Aminohexylgeldanamycin | ||
Aminohexylgeldanamycin (AHGDM), a derivative of Geldanamycin, is a highly effective inhibitor of HSP90. It exhibits considerable antiangiogenic and antitumor properties[1]. | |||
T38522 |
Aminohexylgeldanamycin hydrochloride
AHGDM hydrochloride,Aminohexylgeldanamycin hydrochloride |
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Aminohexylgeldanamycin (AHGDM) hydrochloride is a Geldanamycin derivative and a powerful inhibitor of HSP90. It exhibits significant antiangiogenic and antitumor properties. | |||
T39158 |
17-DMAP-GA
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17-DMAP-GA, a Geldanamycin analogue, acts as an HSP90 inhibitor, leading to cell cycle abnormalities. | |||
T78764 |
Anticancer agent 136
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Apoptosis | Apoptosis |
Anticanceragent 136 (compound 22),一种GDM C17-三唑类似物,对HDF表现出3.38 μM的IC50,与Hsp90有3.86 μM的Kd。本化合物功能为细胞凋亡诱导剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
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T6343 |
Geldanamycin
格尔德霉素,NSC 122750 |
HSP; Influenza Virus; Tyrosine Kinases; Antibacterial; Antibiotic | Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Geldanamycin 是一种 HSP90 抑制剂(Kd:1.2 μM),可特异性破坏糖皮质激素受体 (GR)/HSP 的结合。 |