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Search Results for " geldanamycin "

5

抑制剂 & 化合物

1

天然产物

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Cat. No. Product Name Target Signaling Pathways
T74013 Geldanamycin-FITC

Geldanamycin-FITC 是一种格尔达霉素荧光探针,可用于HSP90抑制剂的荧光偏振分析。Geldanamycin-FITC 也可用于细胞表面HSP90的检测。储存方式:避光。
T37377 Aminohexylgeldanamycin

Aminohexylgeldanamycin (AHGDM), a derivative of Geldanamycin, is a highly effective inhibitor of HSP90. It exhibits considerable antiangiogenic and antitumor properties[1].
T38522 Aminohexylgeldanamycin hydrochloride

AHGDM hydrochloride,Aminohexylgeldanamycin hydrochloride

Aminohexylgeldanamycin (AHGDM) hydrochloride is a Geldanamycin derivative and a powerful inhibitor of HSP90. It exhibits significant antiangiogenic and antitumor properties.
T39158 17-DMAP-GA

17-DMAP-GA, a Geldanamycin analogue, acts as an HSP90 inhibitor, leading to cell cycle abnormalities.
T78764 Anticancer agent 136

Apoptosis Apoptosis
Anticanceragent 136 (compound 22),一种GDM C17-三唑类似物,对HDF表现出3.38 μM的IC50,与Hsp90有3.86 μM的Kd。本化合物功能为细胞凋亡诱导剂。

化合物

Geldanamycin-FITC
Cat.No: T74013
Synonym:
Target:
Aminohexylgeldanamycin
Cat.No: T37377
Synonym:
Target:
Aminohexylgeldanamycin hydrochloride
Cat.No: T38522
Synonym: AHGDM hydrochloride,Aminohexylgeldanamycin hydrochloride
Target:
17-DMAP-GA
Cat.No: T39158
Synonym:
Target:
Anticancer agent 136
Cat.No: T78764
Synonym:
Target: Apoptosis
Cat. No. Product Name Target Signaling Pathways
T6343 Geldanamycin

格尔德霉素,NSC 122750

HSP; Influenza Virus; Tyrosine Kinases; Antibacterial; Antibiotic Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Tyrosine Kinase/Adaptors
Geldanamycin 是一种 HSP90 抑制剂(Kd:1.2 μM),可特异性破坏糖皮质激素受体 (GR)/HSP 的结合。

天然产物

Geldanamycin
Cat.No: T6343
Synonym: 格尔德霉素,NSC 122750
Target: HSP, Influenza Virus, Tyrosine Kinases, Antibacterial, Antibiotic
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