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Cat. No. Product Name Target Signaling Pathways
T3113 Foretinib

GSK089,EXEL-2880,GSK1363089,XL880

VEGFR; Tie-2; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
Foretinib (GSK1363089) 是多靶点酪氨酸激酶抑制剂,能够抑制 Met (IC50:0.4 nM) 和 KDR (IC50:0.9 nM)。
T36246 SJF 8240

c-MET degrader. Comprises MET inhibitor foretinib (GSK 1363089; Cat. No. 6056) joined by a linker to a von Hippel-Lindau (VHL) recruiting ligand. Degrades c-MET within 6 hours in vitro. Inhibits agonist-driven AKT phosphorylation and GTL16 cell proliferation (IC50 = 66.7 nM). Also degrades exon-14-deleted c-MET in Hs746T cells.

化合物

Foretinib
Cat.No: T3113
Synonym: GSK089,EXEL-2880,GSK1363089,XL880
Target: VEGFR, Tie-2, c-Met/HGFR
SJF 8240
Cat.No: T36246
Synonym:
Target:
TargetMol Loading
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