Cat. No. | Product Name | Target | Signaling Pathways |
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TP2022 |
GR231118
GR 231118 |
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Potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively). Also a potent and selective NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 receptors respectively). Suppresses | |||
T75910 |
GR231118 TFA
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GR231118是神经肽Y的C末端类似物,作为人神经肽YY受体的高竞争性和相对选择性的拮抗剂(pKi=10.4),并对人类神经肽Y4受体显示出拮抗效果(pEC50=8.6;pKi=9.6),同时是对人及大鼠神经肽YY2与Y5受体的弱激动剂。此外,GR231118对小鼠神经肽YY6受体具有较高亲和力(pKi=8.8)。 |