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Search Results for " gpr120 "

15

抑制剂 & 化合物

2

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T15413	GPR120 Agonist 3 GPR120-IN-1	GPR	Endocrinology/Hormones; GPCR/G Protein
	GPR120 Agonist 3 (GPR120-IN-1) 是一种有效的、选择性的 Gpr120激动剂，logEC50为 −7.62。
T4312	GPR120 Agonist 2 GPR120 receptor agonist	GPR	Endocrinology/Hormones; GPCR/G Protein
	GPR120 Agonist 2 是一种选择性 GPR120激动剂。
T71862	GPR120-IN-1
	GPR120-IN-1 is a novel GPR120 inhibitor, showing ~90% inhibitory effects on cell growth with micromolar affinities against SW480.
T11454	GPR120 modulator 2	Others	Others
	GPR120 modulator 2 is useful for modulating GPR120.
T11453	GPR120 modulator 1	Others	Others
	GPR120 modulator 1 is useful for modulating GPR120.
T11452	GPR120 Agonist 1	GPR	Endocrinology/Hormones; GPCR/G Protein
	GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GPR120 (the calcium flux assay), respectively.
T22027	AH-7614 AH 7614	GPR	Endocrinology/Hormones; GPCR/G Protein
	AH-7614 (AH 7614) 是一种选择性的游离脂肪酸受体 4(FFA4/GPR120) 拮抗剂，对人和大小鼠 FFA4 的pIC50值分别为 7.1、8.1 和 8.1。它能够阻断多不饱和 ω-6 脂肪酸亚油酸和 FFA4 激动剂的作用。
T1781	GW9508 GW 9508	GPR; Potassium Channel	Endocrinology/Hormones; GPCR/G Protein; Membrane transporter/Ion channel
	GW 9508 是一种选择性 G 蛋白偶联受体FFA1(GPR40) 和GPR120激动剂。它是一种葡萄糖敏感性胰岛素促分泌剂和 ATP 敏感性钾通道开放剂，具有抗炎和抗动脉粥样硬化活性。
TQ0020	AMG 837 calcium hydrate	GPR	Endocrinology/Hormones; GPCR/G Protein
	AMG 837 calcium hydrate 是口服有效的 GPR40/FFA1部分激动剂，抑制 [3H]AMG 837 与人类 FFA1受体的特异性结合，pIC50为 8.13。AMG 837 calcium hydrate 可增强啮齿动物的胰岛素分泌并降低葡萄糖水平。
T22967	MEDICA16 MEDICA 16	GPR; Others; ATP Citrate Lyase	Endocrinology/Hormones; GPCR/G Protein; Metabolism; Others
	MEDICA16 是 GPR40 的特异性激动剂以及 GPR120 的部分激动剂。 MEDICA16 是一种 ATP-柠檬酸裂解酶抑制剂，可显着降低腓肠肌中的细胞内 TG 含量，同时增加胰岛素敏感性。
T3433	TUG-891 TUG 891,TUG891	GPR	Endocrinology/Hormones; GPCR/G Protein
	TUG-891 是一种选择性的长链游离脂肪酸受体 4 (FFA4/GPR120) 的激动剂。
T71194	Metabolex-36
	Metabolex-36 is a selective GPR120 agonist
T28140	NCG21 NCG-21,NCG 21
	NCG21 is a GPR120 agonist, which showed potent extracellular signal-regulated kinase (ERK) activation in a cloned GPR120 system. NCG21 potently activated ERK, intracellular calcium responses and GLP-1 secretion in murine enteroendocrine STC-1 cells that e
T34968	TUG-905
	TUG-905 is an agonist for free fatty acid receptor 4 (FFA4/GPR120), and TUG-905 has the potential to treat agitation.
T36634	ZQ 16
	Selective medium-chain free fatty acid receptor GPR84 agonist (EC50 = 139 nM). Exhibits no response at GPR40, GPR41, GPR119 or GPR120 at 100 μM. Activates calcium mobilization, inhibits cAMP accumulation, and induces ERK1/2 phosphorylation, receptor desensitization and internalization in vitro. Liu et al (2016) Design and synthesis of 2-alkylpyrimidine-4,6-diol and 6-alkylpyridine-2,4-diol as potent GPR84 agonists. ACS Med.Chem.Lett. 7 579 PMID:27326330 \|Zhang et al (2016) Discovery and characte...

化合物

GPR120 Agonist 3

Cat.No: T15413

Synonym: GPR120-IN-1

Target: GPR

GPR120 Agonist 2

Cat.No: T4312

Synonym: GPR120 receptor agonist

Target: GPR

Cat.No: T71862

GPR120 modulator 2

Cat.No: T11454

Target: Others

GPR120 modulator 1

Cat.No: T11453

Target: Others

GPR120 Agonist 1

Cat.No: T11452

Target: GPR

Cat.No: T22027

Synonym: AH 7614

Target: GPR

Cat.No: T1781

Synonym: GW 9508

Target: GPR, Potassium Channel

AMG 837 calcium hydrate

Cat.No: TQ0020

Target: GPR

Cat.No: T22967

Synonym: MEDICA 16

Target: GPR, Others, ATP Citrate Lyase

Cat.No: T3433

Synonym: TUG 891,TUG891

Target: GPR

Cat.No: T71194

Cat.No: T28140

Synonym: NCG-21,NCG 21

Cat.No: T34968

Cat.No: T36634

Cat. No.	Product Name	Target	Signaling Pathways
TN2077	(+/-)-Pinocembrin NSC 43318,(±)-5,7-Dihydroxyflavanone	GPR; Others	Endocrinology/Hormones; GPCR/G Protein; Others
	(+/-)-Pinocembrin (NSC-43318) 是一种来自腋松的天然产物，它是一种 GPR120 配体，能促进 HaCaT 细胞系的伤口愈合。
T3919	Ginsenoside Rb2 Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2	GPR; Others; Influenza Virus; Endogenous Metabolite	Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Others
	Ginsenoside Rb2 (Ginsenoside C) 是人参提取物中的一种主要生物活性成分，具有抗病毒活性，可上调 GPR120 基因表达。

天然产物

(+/-)-Pinocembrin

Cat.No: TN2077

Synonym: NSC 43318,(±)-5,7-Dihydroxyflavanone

Target: GPR, Others

Ginsenoside Rb2

Cat.No: T3919

Synonym: Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2

Target: GPR, Others, Influenza Virus, Endogenous Metabolite

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