Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T15374 |
Ipatasertib dihydrochloride
GDC-0068 dihydrochloride,RG-7440 dihydrochloride |
Akt; PKA | Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors |
Ipatasertib dihydrochloride (GDC-0068 dihydrochloride) 是ATP 竞争性的pan-Akt 选择性抑制剂,抑制Akt1,Akt2,Akt3,IC50分别为 5,18,8 nM。 | |||
T38393 |
Ipatasertib-NH2 dihydrochloride
RG7440-NH2 dihydrochloride,Ipatasertib-NH2 dihydrochloride,GDC-0068-NH2 dihydrochloride |
||
Ipatasertib-NH2 dihydrochloride is a ligand for the target protein AKT in PROTAC INY-03-041. INY-03-041 consists of Ipatasertib-NH2, a ten-hydrocarbon linker, and the CRBN ligand Lenalidomide, which acts as an E3 ubiquitin ligase. |