Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78360 |
Glyceraldehyde phosphate dehydrogenase
GAPDH,G3PDH,GADPH |
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Glyceraldehyde phosphate dehydrogenase是一种酶,既是抗胸腺细胞剂也是抗凋亡剂的靶点,它负责催化过羟基自由基对还原型烟酰胺腺嘌呤二核苷酸(NADH)的链氧化反应。 | |||
T8574 |
SPHINX
|
Others | Others |
SPHINX 是新一代的 SPRK1抑制剂。 | |||
T21792 |
CGP 3466B maleate
马来酸CGP3466B,Omigapil (Maleate),Omigapil maleate |
Apoptosis | Apoptosis |
CGP 3466B maleate (Omigapil maleate) 是一种口服有效的 GAPDH 亚硝基化抑制剂,可消除 Aβ1-42 诱导的小鼠 tau 乙酰化,记忆障碍和运动功能障碍,Omigapil maleate 具有研究阿尔茨海默症的潜力。Omigapil maleate (CGP3446B maleate) 是一种有效的凋亡 (apoptosis) 抑制剂。Omigapil maleate 可用于研究先天性肌营养不良 (CMD)。 | |||
T10966 |
DC-5163
|
Others | Others |
DC-5163 is a potent inhibitor of glyceraldehyde 3-phosphate dehydrogenase (GAPDH) with IC50 of 176.3 nM and Kd of 3.192 μM. DC-5163 selectively inhibits cancer cell proliferation and induces apoptosis, and partially inhibits the glycolysis pathway. | |||
T27735 |
KM05382
KM 05382,KM-05382 |
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KM05382 inhibits CDK9 and the transcription of GAPDH. | |||
T71419 |
Diclazuril K
|
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Diclazuril K is a coccidiostat and GAPDH inhibitor used to prevent parasitic contamination of livestock and poultry feed. | |||
T71418 |
Diclazuril Na
|
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Diclazuril Na is a coccidiostat and GAPDH inhibitor used to prevent parasitic contamination of livestock and poultry feed. | |||
T72879 |
Misetionamide
|
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Misetionamide,一种恶噻嗪类口服化合物,作为甘油醛-3-磷酸脱氢酶 (GAPDH) 抑制剂,展现出抗肿瘤活性,适用于癌症研究。 |