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Cat. No. Product Name Target Signaling Pathways
T62391 FGFR-IN-6

FGFR-IN-6 (Compound 5) 是一种 FGFR 抑制剂。
T2041 PD153035

NSC 669364,SU-5271,ZM 252868,AG1517

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
PD153035 (NSC-669364) 是一种EGFR 抑制剂,Ki 和IC50值分别为6和25 pM。
T2361 LY2874455

LY 2874455,LY-2874455

VEGFR; FGFR Angiogenesis; Tyrosine Kinase/Adaptors
LY2874455 是pan-FGFR 抑制剂,能够抑制FGFR1 (IC50:2.8 nM),FGFR2 (IC50:2.6 nM),FGFR3 (IC50:6.4 nM),FGFR4 (IC50:6 nM)。
T61660 FGFR-IN-3

FGFR-IN-3 (compound 6) is a highly potent and orally active modulator of FGFR (fibroblast growth factor receptor). It has the ability to penetrate the blood-brain barrier (BBB). Additionally, FGFR-IN-3 exhibits significant neuroprotective properties. Therefore, it holds potential for research on neurodegenerative diseases [1].
T82405 FGFR3-IN-6

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
FGFR3-IN-6FGFR3选择性抑制剂,具有低于350 nM 的IC50,适用于癌症研究领域。

化合物

FGFR-IN-6
Cat.No: T62391
Synonym:
Target:
PD153035
Cat.No: T2041
Synonym: NSC 669364,SU-5271,ZM 252868,AG1517
Target: EGFR
LY2874455
Cat.No: T2361
Synonym: LY 2874455,LY-2874455
Target: VEGFR, FGFR
FGFR-IN-3
Cat.No: T61660
Synonym:
Target:
FGFR3-IN-6
Cat.No: T82405
Synonym:
Target: FGFR
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