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Cat. No. Product Name Target Signaling Pathways
T13688 Eribulin

B1939,艾日布林,ER-086526,E7389

Others Others
Eribulin inhibits the proliferation of cancer cells by binding microtubule proteins and microtubules. Eribulin is a microtubule targeting agent that is used in the treatment of metastatic breast cancer.
T13687 Eribulin mesylate

B1939 mesylate,甲磺酸艾日布林,ER-086526 mesylate,E7389 mesylate

Apoptosis; Others; Microtubule Associated Apoptosis; Cytoskeletal Signaling; Others
Eribulin mesylate (E7389 mesylate) 是一种靶向微管的抗癌剂,通过结合微管蛋白和微管来抑制癌细胞的增殖,可研究转移性乳腺癌。
T39579 Mal-(CH2)5-Val-Cit-PAB-Eribulin

Mal-(CH2)5-Val-Cit-PAB-Eribulin

Mal-(CH2)5-Val-Cit-PAB-Eribulin is a potent antitumor ADC drug-linker conjugate that utilizes Eribulin, an anti-microtubule agent, connected through the Mal-(CH2)5-Val-Cit-PAB linker.
T18871 VCP-Eribulin

Others Others
VCP-Eribulin, an Eribulin-based drug for antibody conjugates[1], combines the VCP (ADCs linker) with Eribulin, a distinct microtubule inhibitor used in cancer treatments[2].
T18278 Mal-PEG2-VCP-Eribulin

Others Others
Mal-PEG2-VCP-Eribulin is a chemotherapeutic compound comprising an antibody-drug conjugate (ADC) linker (Mal-PEG2-VCP) and the microtubule inhibitor Eribulin[1]. This compound uniquely targets microtubules, offering a novel approach to cancer treatment. Eribulin is specifically utilized in creating targeted Eribulin-based drugs for antibody conjugates[1].
T82323 GGFG-Eribulin

GGFG-Eribulin(Compound GGFG)是一种用于合成ADCs的ADC-药物连接子偶联物。它由ADC细胞毒素Exatecan和连接子构成,以实现靶向输送药物。
T77908 Farletuzumab ecteribulin

MORAb-202

Farletuzumabecteribulin(MORAb-202)是一款人源化抗人叶酸受体α(FRA)抗体Farletuzumab与Mal-PEG2-Val-Cit-PAB-eribulin通过还原的链间二硫键偶联成的抗体-活性分子偶联物(ADC)。该化合物活性分子抗体比率为4.0,对FRA阳性细胞展示出强大的体外细胞毒性,并具备有效的抗肿瘤活性。

化合物

Eribulin
Cat.No: T13688
Synonym: B1939,艾日布林,ER-086526,E7389
Target: Others
Eribulin mesylate
Cat.No: T13687
Synonym: B1939 mesylate,甲磺酸艾日布林,ER-086526 mesylate,E7389 mesylate
Target: Apoptosis, Others, Microtubule Associated
Mal-(CH2)5-Val-Cit-PAB-Eribulin
Cat.No: T39579
Synonym: Mal-(CH2)5-Val-Cit-PAB-Eribulin
Target:
VCP-Eribulin
Cat.No: T18871
Synonym:
Target: Others
Mal-PEG2-VCP-Eribulin
Cat.No: T18278
Synonym:
Target: Others
GGFG-Eribulin
Cat.No: T82323
Synonym:
Target:
Farletuzumab ecteribulin
Cat.No: T77908
Synonym: MORAb-202
Target:
TargetMol Loading
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