Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7041 |
Donepezil
E2020,Donepezilo,Aricept,多奈哌齐 |
AChE | Neuroscience |
Donepezil (Aricept) 是一种AChE 抑制剂,对牛 AChE 和人 AChE 的IC50分别为 8.12 nM 和 11.6 nM。 | |||
T6478 |
Donepezil Hydrochloride
Aricept,BNAG,E2020,Donepezil HCl,盐酸多奈哌齐 |
AChR; AChE | Neuroscience |
Donepezil HCl(Aricept) 是可逆的选择性AChE 抑制剂,IC50=6.7 nM,对 AChE 的选择性高于 BuChE。Donepezil Hydrochloride (Aricept) 对 Aβ42 神经毒性具有神经保护作用。 | |||
T61638 |
Dihydro Donepezil
|
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Dihydro Donepezil, also known as Dihydro E2020, is a metabolite derived from Donepezil. Donepezil is a highly specific and potent inhibitor of acetylcholinesterase (AChE) with IC50 values of 8.12 nM and 11.6 nM for butyrylcholinesterase (bAChE) and human acetylcholinesterase (hAChE), respectively [1]. |