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Cat. No. Product Name Target Signaling Pathways
T6364 Desfesoterodine

5-HMT,(R)-5-Hydroxymethyl Tolterodine,(R)-5-羟甲基托特罗定,PNU-200577,5-HM,5-hydroxymethyl Tolterodine

AChR Neuroscience
Desfesoterodine (5-HMT) 是选择性毒蕈碱受体拮抗剂,Kb 和pA2分别为 0.84 nM 和 9.14。它可改善大鼠脑梗死诱导膀胱过度活动,是 Tolterodine 和 Fesoterodine 的主要药理活性代谢产物。
T31238 DE(isopropyl)desfesoterodine

N-Desisopropyl desfesoterodine

DE(isopropyl)desfesoterodine is a biochemical.
T6364L Desfesoterodine fumarate

PNU-200577 fumarate,UNII-607O3D83YQ

Desfesoterodine fumarate is a bio-active chemical. Detailed information has not been published.
T40161 (Rac)-5-Hydroxymethyl Tolterodine hydrochloride

(Rac)-5-Hydroxymethyl Tolterodine hydrochloride,(Rac)-PNU-200577hydrochloride,(Rac)-Desfesoterodine hydrochloride

(Rac)-5-Hydroxymethyl Tolterodine hydrochloride, also known as (Rac)-Desfesoterodine hydrochloride, is an active metabolite of Tolterodine that functions as a mAChR antagonist. It exhibits significant affinity (K i values) for M1, M2, M3, M4, and M5 receptors, with values of 2.3 nM, 2 nM, 2.5 nM, 2.8 nM, and 2.9 nM, respectively. This compound is commonly employed in research related to overactive bladder conditions.
T9419 Fesoterodine

(R) Fesoterodine,弗斯特罗定

AChR Neuroscience
Fesoterodine ((R) Fesoterodine) 是可口服的,非亚型选择性的竞争性毒蕈碱受体拮抗剂,用于膀胱过度活动症,对 M1、M2、M3、M4 和 M5 受体的pKi 值分别为 8.0、7.7、7.4、7.3 和 7.5。
T1475 Fesoterodine fumarate

Toviaz,SPM 907,富马酸非索罗定

AChR Neuroscience
Fesoterodine fumarate (Toviaz) 是可口服的,非亚型选择性的竞争性毒蕈碱受体拮抗剂,用于膀胱过度活动症,对 M1、M2、M3、M4 和 M5 受体的pKi 值分别为 8.0、7.7、7.4、7.3 和 7.5。

化合物

Desfesoterodine
Cat.No: T6364
Synonym: 5-HMT,(R)-5-Hydroxymethyl Tolterodine,(R)-5-羟甲基托特罗定,PNU-200577,5-HM,5-hydroxymethyl Tolterodine
Target: AChR
DE(isopropyl)desfesoterodine
Cat.No: T31238
Synonym: N-Desisopropyl desfesoterodine
Target:
Desfesoterodine fumarate
Cat.No: T6364L
Synonym: PNU-200577 fumarate,UNII-607O3D83YQ
Target:
(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
Cat.No: T40161
Synonym: (Rac)-5-Hydroxymethyl Tolterodine hydrochloride,(Rac)-PNU-200577hydrochloride,(Rac)-Desfesoterodine hydrochloride
Target:
Fesoterodine
Cat.No: T9419
Synonym: (R) Fesoterodine,弗斯特罗定
Target: AChR
Fesoterodine fumarate
Cat.No: T1475
Synonym: Toviaz,SPM 907,富马酸非索罗定
Target: AChR
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