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Search Results for " dhp "

19

抑制剂 & 化合物

3

天然产物

3

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T27164	DHP-218 PAK-9,PAK9,PAK 9,DHP218
	DHP-218 is a calcium channel antagonist. DHP-218 inhibits Calcium-induced contraction of the rat aorta in high K+ solution with the pA2 value of 9.11. The IC50 value for the inhibitory effects of DHP-218 in high K+-induced and phenylephrine-induced contra
T36912	17α,20β-Dihydroxy-4-pregnen-3-one 17α,20β-dihydroxy Progesterone,17α,20β-DHP,17α,20β-Dihydroxy-4-pregnen-3-one
	17α,20β-Dihydroxy-4-pregnen-3-one (17α,20β-DHP) is an endogenous, maturation-inducing steroid that stimulates oocyte maturation in females of several teleost species. For example, 1 μg/ml of 17α,20β-DHP applied to Persian sturgeon oocytes has been shown to effectively induce germinal vesicle breakdown, an essential step during oocyte maturation.1 Gonadotropin-releasing hormone and the gonadotropins, follicle-stimulating hormone and luteinizing hormone, have been shown to stimulate the production...
T12004	Meropenem trihydrate 美罗培南三水合物,SM 7338 trihydrate	Antibacterial; Antibiotic	Microbiology/Virology
	Meropenem trihydrate (SM 7338 trihydrate) 是一种碳青霉烯抗生素，具有广谱抗菌活性。它对敏感和耐药的杜克氏杆菌 (MIC 值为 0.015-0.12 mg/mL)，淋病奈瑟氏球菌 (MIC 值为 0.02-0.06 mg/mL)和流感嗜血杆菌 (MIC 值为 0.03-0.12 mg/mL) 具有活性。
T11032	DHPG (RS)-3,5-DHPG,DL-Α-(3,5-二羟基苯基)甘氨酸	GluR	Neuroscience
	DHPG ((RS)-3,5-DHPG) 是一种氨基酸，是选择性代谢型谷氨酸受体 mGluR 的激动剂，也是与磷脂酶 D 耦合的 mGluR 的有效拮抗剂。
T18912	ADHP 10-乙酰基-3,7-二羟基吩嗪,10-Acetyl-3,7-dihydroxyphenoxazine	Others	Others
	ADHP (10-Acetyl-3,7-dihydroxyphenoxazine) 是荧光过氧化物酶底物，其λex=530 nm，λem=590 nm。
T83938	TAT-PDHPS1
	TAT-PDHPS1是一种针对Yes-associated protein (YAP) 信号的肽抑制剂。它由内源性肽PDHPS1和能穿透细胞的肽序列TAT组成。PDHPS1与蛋白磷酸酶2磷酸酶激活因子(PTPA)结合, 激活蛋白磷酸酶2A (PP2A)。该激活促进YAP的磷酸化和抑制YAP靶向基因的表达。TAT-PDHPS1能够抑制体外卵巢癌细胞的增殖和小鼠皮下异种移植肿瘤模型中的卵巢肿瘤生长。
T40275	DHPS-IN-1
	DHPS-IN-1, a chemical compound, demonstrates exceptional inhibitory potency against melanoma cells, as evidenced by its IC50 value of 0.014 μM.
T25318	DHPCC-9 DHPCC9
	DHPCC-9 is an inhibitor of Pim kinase.
T23289	(S)-3,5-DHPG	Others	Others
	group I mGlu receptor agonist
T70684	DHPM-93
	DHPM-93 is a the most potent inhibitor of sodium iodide symporter (nis) reported to date
T23988	DHPCG
	DHPCG is an inhibitor of HIF-1α prolyl hydroxylase.
T0112L	Diltiazem Diltiazem free base,Dilticard,地尔硫卓,CRD-401,CRD401,Dilzen,CRD 401
	Diltiazem is a non-dihydropyridine (non-DHP) calcium channel blocker that relaxes the smooth muscle in arterial walls, thus opening (dilating) arteries, allowing easier blood flow, and lowering blood pressure, and is used to treat hypertension, angina pec
T24932	Vatanidipine AE-0047,AE 0047,AE0047	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Vatanidipine (AE0047) 是一种新型的双氢吡啶(DHP)型钙通道阻滞剂，具有缓慢起效的药理作用。在各种实验性高血压模型中观察到缓慢起效和持久的降压作用。
T37319	5β-Dihydroprogesterone
	5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHP inhibits spontaneous contractions in isolated rat uterus when used at a concentration of 10 μg/ml, an effect that can be blocked by the progesterone receptor antagonist RU486 but not the GABAAreceptor antagonist picrotoxin .1It is a negative modulator of homooligomeric Ρ1 subunit-containing GABAAreceptors, inhibiting GABA-induced currents in...
T34483	Sadopine
	Sadopine is an excellent high affinity, high specific activity radioligand to label selectively the DHP receptor of L-type Ca2+ channels in tissue sections as well as in membrane fragments.
T23710	Watanidipine dihydrochloride
	Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.
T66029	3,4-Dehydro-L-proline
	The leguminous shrub,Leucaena leucocephala(Leucaena) is wide‐spread in tropical and subtropical agricultural systems and provides a ready source of protein for livestock. However, the presence of mimosine, a non‐protein, amino acid comprising about 12% of the dry matter in growing tips ofLeucaena, is toxic to animals. Mimosine is degraded rapidly in the rumen to produce 3,4‐dihydroxypyridine (3,4‐DHP) and 2,3‐dihydroxypyridine (2,3‐DHP), both of which remain toxic to animals[1]. 3,4-DHP, as a de...
T79605	RIP1 kinase inhibitor 8	Necroptosis	Apoptosis
	RIP1 kinase inhibitor 8（Compound 77）是一种高选择性的二氢吡唑（DHP）RIP1激酶抑制剂，其IC50值为20 nM，可有效抑制坏死（necrotic）细胞死亡，并在多种物种中展现出优良的药代动力学属性。
T60649	AV-153 free base
	AV-153 free base 是一种 1,4-二氢吡啶(1,4-DHP) 衍生物。AV-153 free base 是一种抗诱变剂，具有抗癌活性。AV-153 free base 可以与胞嘧啶和胸腺嘧啶相互作用，并影响聚 (ADP) 核糖基化。在体外实验中，AV-153 free base 在 DNA 的单链断裂处插入到 DNA 并减少 DNA 损伤，刺激 DNA 修复。

化合物

Cat.No: T27164

Synonym: PAK-9,PAK9,PAK 9,DHP218

17α,20β-Dihydroxy-4-pregnen-3-one

Cat.No: T36912

Synonym: 17α,20β-dihydroxy Progesterone,17α,20β-DHP,17α,20β-Dihydroxy-4-pregnen-3-one

Meropenem trihydrate

Cat.No: T12004

Synonym: 美罗培南三水合物,SM 7338 trihydrate

Target: Antibacterial, Antibiotic

Cat.No: T11032

Synonym: (RS)-3,5-DHPG,DL-Α-(3,5-二羟基苯基)甘氨酸

Target: GluR

Cat.No: T18912

Synonym: 10-乙酰基-3,7-二羟基吩嗪,10-Acetyl-3,7-dihydroxyphenoxazine

Target: Others

Cat.No: T83938

Cat.No: T40275

Cat.No: T25318

Synonym: DHPCC9

Cat.No: T23289

Target: Others

Cat.No: T70684

Cat.No: T23988

Cat.No: T0112L

Synonym: Diltiazem free base,Dilticard,地尔硫卓,CRD-401,CRD401,Dilzen,CRD 401

Cat.No: T24932

Synonym: AE-0047,AE 0047,AE0047

Target: Calcium Channel

5β-Dihydroprogesterone

Cat.No: T37319

Cat.No: T34483

Watanidipine dihydrochloride

Cat.No: T23710

3,4-Dehydro-L-proline

Cat.No: T66029

RIP1 kinase inhibitor 8

Cat.No: T79605

Target: Necroptosis

AV-153 free base

Cat.No: T60649

Cat. No.	Product Name	Target	Signaling Pathways
T0224	Meropenem 美罗培南,SM 7338	Others; Antibacterial; Antibiotic	Microbiology/Virology; Others
	Meropenem (SM 7338) 是一种具有广谱抗菌活性的碳青霉烯抗生素，对敏感和耐药的淋病奈瑟氏球菌，流感嗜血杆菌和杜克氏杆菌的 MIC 值分别为 0.02-0.06 mg/mL，0.03-0.12 mg/mL 和 0.015-0.12 mg/mL。
T74193	(R)-IDHP
	(R)-IDHP为IDHP异构体，属于丹参代谢物。该化合物能通过抑制血管平滑肌细胞电压依赖性钙通道与受体操作钙通道的Ca2+释放和Ca2+内流，发挥血管松弛作用，适用于心脑血管疾病研究。
TN3118	5-Hydroxy-7-(4'-hydroxy-3'-methoxyphenyl)-1-phenyl-3-heptanone (DHPA)	Others	Others
	5-Hydroxy-7-(4'-hydroxy-3'-methoxyphenyl)-1-phenyl-3-heptanone (DHPA) is a pancreatic lipase inhibitor, it shows antihyperlipidemic activity.

天然产物

Cat.No: T0224

Synonym: 美罗培南,SM 7338

Target: Others, Antibacterial, Antibiotic

Cat.No: T74193

5-Hydroxy-7-(4'-hydroxy-3'-methoxyphenyl)-1-phenyl-3-heptanone (DHPA)

Cat.No: TN3118

Target: Others

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-03791	DPYS Protein, Human, Recombinant dihydropyrimidinase,DHPase,DHP	Human	Baculovirus Insect Cells
	DPYS Protein, Human, Recombinant is expressed in Baculovirus insect cells. The predicted molecular weight is 56.8 kDa and the accession number is Q14117.
TMPY-03790	DPYS Protein, Human, Recombinant (His & GST) DHPase,dihydropyrimidinase,DHP	Human	Baculovirus Insect Cells
	DPYS Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 84.4 kDa and the accession number is Q14117.
TMPJ-01374	UPB1 Protein, Human, Recombinant (His) β-Ureidopropionase,Beta-Alanine Synthase,β-Alanine Synthase,...	Human	E. coli
	β-Ureidopropionase is a cytoplasmic protein which belongs to the CN hydrolase family of BUP subfamily. β-Ureidopropionase binds one zinc ion per subunit, catalyzes the last step in the pyrimidine degradation pathway. β-Ureidopropionase can convert N-carbamyl-beta-aminoisobutyric acid and N-carbamyl-beta-alanine to beta-aminoisobutyric acid and beta-alanine, ammonia and carbon dioxide, respectively. The pyrimidine bases uracil and thymine are degraded via the consecutive action of dihydropyrimidi...

重组蛋白

DPYS Protein, Human, Recombinant

Cat.No: TMPY-03791

Species: Human

Expression System: Baculovirus Insect Cells

DPYS Protein, Human, Recombinant (His & GST)

Cat.No: TMPY-03790

Species: Human

Expression System: Baculovirus Insect Cells

UPB1 Protein, Human, Recombinant (His)

Cat.No: TMPJ-01374

Species: Human

Expression System: E. coli

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