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Cat. No. Product Name Target Signaling Pathways
T11044 Dihydromunduletone

DHM

GPR Endocrinology/Hormones; GPCR/G Protein
Dihydromunduletone (DHM) 是一种粘附 G 蛋白偶联受体 (aGPCR)拮抗剂,可做一种化学探针,对具有相似拴系激动剂的 GPR56 和 GPR114/ADGRG5 有抑制作用。
T21252 DHMB

2,3-Dihydroxy-4-Methoxybenzaldehyde

Others Others
DHMB (2,3-Dihydroxy-4-Methoxybenzaldehyde) 对肠上皮细胞发挥保护作用。 DHMB 具有抗炎和抗真菌能力。
T13462 (+)-DHMEQ

(1R,2R,6R)-Dehydroxymethylepoxyquinomicin,(1R,2R,6R)-DHMEQ

Others Others
(+)-DHMEQ is an antioxidant transcription factor Nrf2 activator. (+)-DHMEQ is the enantiomer of (-)-DHMEQ.
T11018 DHMEQ racemate

rel-DHMEQ

NF-κB NF-κB
DHMEQ racemate is an NF-κB inhibitor. The activity of DHMEQ racemate is lower than (-)-DHMEQ.
T27162 DHMPA

DHMPA is an inhibitor of catechol-O-methyltransferase (COMT), it also reduces tissue norepinephrine and blood pressure.

化合物

Dihydromunduletone
Cat.No: T11044
Synonym: DHM
Target: GPR
DHMB
Cat.No: T21252
Synonym: 2,3-Dihydroxy-4-Methoxybenzaldehyde
Target: Others
(+)-DHMEQ
Cat.No: T13462
Synonym: (1R,2R,6R)-Dehydroxymethylepoxyquinomicin,(1R,2R,6R)-DHMEQ
Target: Others
DHMEQ racemate
Cat.No: T11018
Synonym: rel-DHMEQ
Target: NF-κB
DHMPA
Cat.No: T27162
Synonym:
Target:
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