Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11044 |
Dihydromunduletone
DHM |
GPR | Endocrinology/Hormones; GPCR/G Protein |
Dihydromunduletone (DHM) 是一种粘附 G 蛋白偶联受体 (aGPCR)拮抗剂,可做一种化学探针,对具有相似拴系激动剂的 GPR56 和 GPR114/ADGRG5 有抑制作用。 | |||
T21252 |
DHMB
2,3-Dihydroxy-4-Methoxybenzaldehyde |
Others | Others |
DHMB (2,3-Dihydroxy-4-Methoxybenzaldehyde) 对肠上皮细胞发挥保护作用。 DHMB 具有抗炎和抗真菌能力。 | |||
T13462 |
(+)-DHMEQ
(1R,2R,6R)-Dehydroxymethylepoxyquinomicin,(1R,2R,6R)-DHMEQ |
Others | Others |
(+)-DHMEQ is an antioxidant transcription factor Nrf2 activator. (+)-DHMEQ is the enantiomer of (-)-DHMEQ. | |||
T11018 |
DHMEQ racemate
rel-DHMEQ |
NF-κB | NF-κB |
DHMEQ racemate is an NF-κB inhibitor. The activity of DHMEQ racemate is lower than (-)-DHMEQ. | |||
T27162 | DHMPA | ||
DHMPA is an inhibitor of catechol-O-methyltransferase (COMT), it also reduces tissue norepinephrine and blood pressure. |