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Cat. No. Product Name Target Signaling Pathways
T13349 WS-383

E1/E2/E3 Enzyme Ubiquitination
WS-383 是高效、选择性、可逆的DCN1-UBC12相互作用抑制剂,IC50为11 nM。它抑制 Cul3/1 的类泛素化修饰,引起 NRF2,p21和p27 的积累。
T63647 DCN1-UBC12-IN-1

DCN1-UBC12-IN-1 是有效的、特异性的 DCN1-UBC12 抑制剂,其 IC50 值为 2.86 nM,具有抗心脏成纤维化活性。
T63820 DCN1-UBC12-IN-2

DCN1-UBC12-IN-2 是有效的、特异性的 DCN1-UBC12 抑制剂,其 IC50 值为 9.55 nM。DCN1-UBC12-IN-2 能够特异性靶向 DCN1-UBC12 相互作用,减缓 Ang II 诱导的心脏成纤维细胞活化。
T9140 NAcM-OPT HCl(2089293-61-6 free base)

NEDD8 Metabolism
NAcM-OPT HCl(2089293-61-6 free base) 是一种可口服的 cullin neddylation 1 (DCN1) 抑制剂,靶向 N-Acetyl-UBE2M(E2 结合酶,UBC12)与 DCN1 的相互作用,IC50 为 79 nM。
T13348 WS-383 free base

Others Others
WS-383 free base is a selective and reversible DCN1-UBC12 interaction inhibitor(IC50 of 11 nM).
T11033 DI-591

Others Others
DI-591 is an effective, high-affinity and cell-permeability inhibitor for DCN1-UBC12 interaction. DI-591 binds to DCN1 and DCN2 with Ki values of 12 and nM and 10.4 nM, respectively, and has no obvious binding to DCN3, DCN4 and DCN5 proteins.
T23989 DI-404

DI-404 is a high-Affinity Peptidomimetic the DCN1-UBC12 Protein-Protein Interaction inhibitor (Kd= 6.9 nM). DI-404 effectively and selectively inhibits the neddylation of cullin 3 over other cullin members.

化合物

WS-383
Cat.No: T13349
Synonym:
Target: E1/E2/E3 Enzyme
DCN1-UBC12-IN-1
Cat.No: T63647
Synonym:
Target:
DCN1-UBC12-IN-2
Cat.No: T63820
Synonym:
Target:
NAcM-OPT HCl(2089293-61-6 free base)
Cat.No: T9140
Synonym:
Target: NEDD8
WS-383 free base
Cat.No: T13348
Synonym:
Target: Others
DI-591
Cat.No: T11033
Synonym:
Target: Others
DI-404
Cat.No: T23989
Synonym:
Target:
TargetMol Loading
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