Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78779 |
D3R/MOR antagonist 2
|
Dopamine Receptor | GPCR/G Protein; Neuroscience |
D3R/MOR antagonist 2(Compound 121)为一种D3R/MOR拮抗剂,其Ki值分别为46.5 nM及691 nM。该化合物通过MOR部分激动作用可产生镇痛效果,并通过D3R拮抗减少阿片类药物的潜在滥用风险。 | |||
T79547 |
MOR agonist-2
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
MOR agonist-2 (Compound 46) 为D3R拮抗剂及MOR激动剂,其Ki值分别为7.26 nM和564 nM。MOR agonist-2潜在以MOR部分激动机制实现镇痛效果,并通过D3R拮抗降低阿片类药物的滥用风险。 |