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Cat. No. | Product Name | Target | Signaling Pathways |
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T76170 | D-Amino acid oxidase | ||
D-Amino acid oxidase 是一种酶,主要负责在动物体内代谢外源性 D-氨基酸以进行解毒,并能够调节大脑中D-丝氨酸的水平。 | |||
T7476 |
AS057278
3-Methylpyrazole-5-carboxylic acid,5-甲基-1H-吡唑-3-羧酸 |
Others | Others |
AS057278 (3-Methylpyrazole-5-carboxylic acid) 是一种 D-氨基酸氧化酶 (DAAO) 抑制剂。 | |||
T38863 |
Luvadaxistat
TAK-831,Luvadaxistat |
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TAK-831 is a potent and highly selective inhibitor of D-amino acid oxidase (DAAO), offering great potential for utilization in schizophrenia research. | |||
T5206 |
DAAO inhibitor-1
|
Others | Others |
DAAO inhibitor-1是 D-氨基酸氧化酶抑制剂(IC50:0.12 μM)。 | |||
T8124 |
Sodium benzoate
Benzoic acid sodium salt,苯甲酸钠 |
Others | Others |
Sodium benzoate (Benzoic acid sodium salt) 是一种 D-氨基酸氧化酶抑制剂。它是一种食品防腐剂。 | |||
T28964 |
Thiolactomycin
|
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Thiolactomycin is a novel reversible dual inhibitor of D-amino acid oxidase (DAO) and D-Aspartate oxidase (DDO). | |||
T78231 | DAO-IN-1 | Others | Others |
DAO-IN-1是高效的D-氨基酸氧化酶(DAO)抑制剂,其IC50值为269 nM。DAO负责d-丝氨酸的代谢,而d-丝氨酸是NMDA受体的共激动剂。 | |||
T37605 |
D-DOPA
|
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D-DOPA is an enantiomer of the dopamine precursor L-DOPA . It can be converted to L-DOPAviasequential oxidation and transamination, which are mediated by D-amino acid oxidase (DAAO) and DOPA transaminase, respectively, in rat kidney homogenates.1It reduces the number of dopaminergic neurons in primary rat embryonic mesencephalic cultures in a concentration-dependent manner.2Intraventricular administration of D-DOPA (200 μg/animal) increases striatal dopamine levels in rats.3D-DOPA (20 mg/kg, i.p... |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10933 |
D-Cysteine
|
Endogenous Metabolite; Antibacterial | Metabolism; Microbiology/Virology |
D-Cysteine 是一种大肠杆菌生长的有力抑制剂,是半胱氨酸的 D 型异构体。它由 D-氨基酸氧化酶介导产生 H2S,是一种对抗小脑共济失调的神经保护剂。 D-半胱氨酸可以抑制由变形链球菌和链球菌血红蛋白形成的两种生物膜的生长和致龋性。 | |||
T19302 |
D(-)-2-Aminobutyric acid
|
Endogenous Metabolite | Metabolism |
D(-)-2-Aminobutyric acid 是一种 D-氨基酸氧化酶的底物。 | |||
T4716 |
Pyrrole-2-carboxylic acid
吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline |
Endogenous Metabolite | Metabolism |
Pyrrole-2-carboxylic acid (Minaline) 是一种天然生物碱类,从海洋细菌Pelomonas puraquaesp. Nov 中分离得到。 | |||
T10938 |
D-Kynurenine
D-尿嘧啶,(R)-2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid,ZINC901103 |
GPR; AhR; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism |
D-Kynurenine (ZINC901103) 是 D-色氨酸的代谢物和 GPR109B 的激动剂。 D-Kynurenine 激活 AhR 并促进上皮细胞向间充质的转化。 D-Kynurenine 在 D-氨基酸氧化酶的荧光分析中用作底物。 |