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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T126510 Crebanine N-oxide

Crebanine N-oxide 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126510,CAS号为 102719-85-7。

化合物

Crebanine N-oxide
Cat.No: T126510
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2S2215 Crebanine

Apoptosis; Others; Akt Apoptosis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling
Crebanine 是来自于韦诺萨千金藤的一种生物碱,通过抑制 MAPKs 和 Akt 信号通路表现出抗炎活性,还具有抗心律失常的作用。它可诱导人类癌细胞的 G1阻滞和凋亡。
TN3799 Dehydrocrebanine

Antifection Microbiology/Virology
Dehydrocrebanine has strong activity against promyelocytic leukemia cells (HL-60) with an IC50 of 2.14 ug/mL. It also shows potent antimalarial activity with an IC50 value of 70 ng/ml.
T81587 Oxocrebanine

Oxocrebanine, 阿朴啡类生物碱,Fissistigma poilanei(番荔枝科)所含。
TN5061 Stephanine

Adrenergic Receptor; Antifection GPCR/G Protein; Microbiology/Virology; Neuroscience
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of 6.76. Stephanine shows significant antiplasmodial activities with IC(50) ranged from 1.2 uM to 52.3 uM. Stephanine and crebanine have high inhibitory activity against gram-positive animal pathogenic bacteria, with MIC values of 0.078-0.312g/l, but low inhibitory activity against gram-negative animal pathogenic bacteria, they also inhibit...

天然产物

Crebanine
Cat.No: T2S2215
Synonym:
Target: Apoptosis, Others, Akt
Dehydrocrebanine
Cat.No: TN3799
Synonym:
Target: Antifection
Oxocrebanine
Cat.No: T81587
Synonym:
Target:
Stephanine
Cat.No: TN5061
Synonym:
Target: Adrenergic Receptor, Antifection
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