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Cat. No. Product Name Target Signaling Pathways
T6322 Copanlisib

BAY 80-6946,可泮利塞,库潘尼西

Apoptosis; PI3K Apoptosis; PI3K/Akt/mTOR signaling
Copanlisib (BAY 80-6946) 是一种选择性的和 ATP 竞争性的泛 I 类PI3K 抑制剂,具有抗肿瘤活性,对PI3Kα,PI3Kδ,PI3Kβ和PI3Kγ的IC50分别为 0.5 nM、0.7 nM、3.7 nM 和 6.4 nM。
T14998 Copanlisib dihydrochloride

库潘尼西盐酸,BAY 80-6946 dihydrochloride

Apoptosis; PI3K; mTOR Apoptosis; PI3K/Akt/mTOR signaling
Copanlisib dihydrochloride (BAY 80-6946 dihydrochloride) 是一种选择性和 ATP 竞争性的泛 I 类 PI3K 抑制剂。它具有优越的抗肿瘤活性,对除 mTOR 以外的其他脂质和蛋白激酶的选择性也超过 2,000 倍。
T70758 Copanlisib HCl hydrate

Copanlisib Dihydrochloride is a novel phosphoinositide 3-kinase (pi3k) inhibitor, inhibiting the activation of the pi3k signaling pathway, resulting in inhibition of tumor cell growth and survival in susceptible tumor cell populations
T70756 KT172

KT172 是一种 DAGLβ抑制剂,IC50值为 11 nM。KT172 可用于代谢和炎症的研究。
T35534 7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine

7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine is a building block.1It has been used in the synthesis of PI3K inhibitors. 1.Scott, W.J., Hentemann, M.F., Rowley, R.B., et al.Discovery and SAR of novel 2,3-dihydroimidazo[1,2-c]quinazoline PI3K inhibitors: Identification of copanlisib (BAY 80-6946)ChemMedChem.11(14)1517-1530(2016)

化合物

Copanlisib
Cat.No: T6322
Synonym: BAY 80-6946,可泮利塞,库潘尼西
Target: Apoptosis, PI3K
Copanlisib dihydrochloride
Cat.No: T14998
Synonym: 库潘尼西盐酸,BAY 80-6946 dihydrochloride
Target: Apoptosis, PI3K, mTOR
Copanlisib HCl hydrate
Cat.No: T70758
Synonym:
Target:
KT172
Cat.No: T70756
Synonym:
Target:
7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine
Cat.No: T35534
Synonym:
Target:
TargetMol Loading
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