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Cat. No. Product Name Target Signaling Pathways
T14983 Clomethiazole

Distraneurin,Chlormethiazole,氯美噻唑,5-(2-CHLOROETHYL)-4-METHYLTHIAZOLE

P450; GABA Receptor Membrane transporter/Ion channel; Metabolism; Neuroscience
Clomethiazole (Distraneurin) 是口服GABAA 激动剂,可抑制人肝微粒体中的细胞色素 P450 异构体,CYP2A6 和 CYP2E1。它有抗惊厥作用,具有治疗惊厥性癫痫持续状态的潜力。
T10796 Chlormethiazole hydrochloride

氯美噻唑盐酸盐,Clomethiazole hydrochloride

Others Others
Chlormethiazole hydrochloride 是抗惊厥药。它具有神经保护作用,能够阻碍 MDMA 诱导的血清素能神经末梢退化。
T27007 Chlormethiazole edisylate

Clomethiazole ethanedisulfonate,Clomethiazole edisylate,Heminevrin,Hemithiamine,Distraneurin

Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.

化合物

Clomethiazole
Cat.No: T14983
Synonym: Distraneurin,Chlormethiazole,氯美噻唑,5-(2-CHLOROETHYL)-4-METHYLTHIAZOLE
Target: P450, GABA Receptor
Chlormethiazole hydrochloride
Cat.No: T10796
Synonym: 氯美噻唑盐酸盐,Clomethiazole hydrochloride
Target: Others
Chlormethiazole edisylate
Cat.No: T27007
Synonym: Clomethiazole ethanedisulfonate,Clomethiazole edisylate,Heminevrin,Hemithiamine,Distraneurin
Target:
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