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Cat. No.	Product Name	Target	Signaling Pathways
T38931	Calpain Inhibitor-1
	Calpain Inhibitor-1 (compound 36) is a highly potent and selective inhibitor of Calpain 1 (Cal1), which is a cysteine protease. It exhibits an IC50 value of 100 nM and a Ki value of 2.89 μM.
T6583	MG-101 ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I	Cysteine Protease; Proteasome	Proteases/Proteasome; Ubiquitination
	MG-101 (Calpain inhibitor I) 是一种有效的半胱氨酸蛋白酶抑制剂，能够抑制钙蛋白酶I (Ki:190 pM)，钙蛋白酶II (Ki:220 pM)，组织蛋白酶B (Ki:150 pM)和组织蛋白酶L (Ki:500 pM)。
T9710	Dazcapistat	Cysteine Protease	Proteases/Proteasome
	Dazcapistat 是一种有效的 calpain 抑制剂，对 calpain 1、calpain 2 和 calpain 9 的 IC50 值均 <3 μM。
T2493	PD 151746	Cysteine Protease; Proteasome	Proteases/Proteasome; Ubiquitination
	PD151746 is a calpain inhibitor with a 20-fold selectivity for u-calpain (Ki = 0.26 ± 0.03 μM) over m-calpain (Ki = 5.33 ± 0.77 μM). Its IC50 values are 0.26 ± 0.03 μM (Ki for μ-calpain) and 5.33 ± 0.77 μM (Ki for m-calpain) [1]. In vitro, PD151746 targets calpain and reduces oxLDL-induced cytotoxicity [2].
T72439	Calpain Inhibitor XI
	Calpain Inhibitor XI，一种可逆的calpain-1共价抑制剂，适用于神经退行性疾病的研究。
T63708	Calpain-2-IN-1
	Calpain-2-IN-1是选择性的钙蛋白酶-2抑制剂，能够延长 ERK 激活，进而增强学习和记忆。
T13486	Neurodegenerative Disorder-Targeting Compound 1	Others	Others
	Neurodegenerative Disorder-Targeting Compound 1 是一种靶向 calpain 的抑制剂。
T14187	ALLM Calpain inhibitor II	Others	Others
	ALLM (Calpain inhibitor II), a potent calpain and cathepsin protease inhibitor, not only prevents neuronal cell death but also enhances chronic neurological function following spinal cord injury (SCI)[1][2].
T28786	SJA6017 SJA-6017,Calpain Inhibitor VI,Calpain-In-4,SJA 6017,Calpain Inhibitor 4
	SJA6017 is a inhibitor of calpain-1 (IC50 = 7.5 nM) and calpain-2 ( IC50 = 78 nM). SJA6017 also inhibits cathepsins B (IC50s = 15 nM) and cathepsins L (IC50s = 1.6 nM). SJA6017 reduces apoptotic cell death, preserves spinal cord tissue and improves functi
T80551	Calpain inhibitor V Mu-Val-HPh-FMK	Antibiotic	Microbiology/Virology
	Calpain inhibitor V (Mu-Val-HPh-FMK) 为具抗衣原体活性的细胞渗透性不可逆钙蛋白酶抑制剂。
T80103	Z-Leu-Tyr-Chloromethylketone
	Z-Leu-Tyr-Chloromethylketone是一种抑制剂，专门针对钙蛋白酶(calpain)活性。
T78632	Z-LLY-FMK Calpain Inhibitor IV	Proteasome	Proteases/Proteasome; Ubiquitination
	Z-LLY-FMK (Calpain Inhibitor IV) 为一种钙蛋白酶抑制剂，涉及调控多个细胞系统的凋亡过程。该化合物能够抑制胆总管结扎所引起的肠细胞凋亡(apoptosis)。
T83527	(Rac)-Neurodegenerative Disorder-Targeting Compound 1
	(Rac)-Neurodegenerative Disorder-Targeting Compound 1为一种针对神经退行性疾病的化合物，具有calpain抑制活性。
T21949	Calpain Inhibitor XII
	(Rac)-Calpain Inhibitor XII是一种可逆的，选择性抑制钙蛋白酶I（calpain I; μ-calpain）的化合物，具有19 nM的Ki值。其对钙蛋白酶II（calpain II; m-calpain; Ki=120 nM）和组织蛋白酶B（cathepsin B; Ki=750 nM）显示出较低的抑制亲和力。(Rac)-Calpain Inhibitor XII用于研究钙蛋白酶在多种生理过程中的角色，如嗜中性粒细胞趋化性、神经元信号传导和心脏对损伤的响应。
T75794	Acetyl-Calpastatin(184-210)(human) TFA
	Acetyl-Calpastatin(184-210)(human) TFA 是一种有效，选择性和可逆的钙蛋白酶 (calpain) 抑制剂，对 μ-钙蛋白酶和组织蛋白酶 L 的Ki 值分别为 0.2 nM 和 6 μM。
T76364	Ac-Leu-Leu-Norleucinol
	Ac-Leu-Leu-Norleucinol 是钙蛋白酶抑制剂，可用于研究对 Acetaminophen 引起的急性肝损伤，并能够降低诱导引发的谷草转氨酶 (ALT) 和谷丙转氨酶 (AST) 水平。

化合物

Calpain Inhibitor-1

Cat.No: T38931

Cat.No: T6583

Synonym: ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I

Target: Cysteine Protease, Proteasome

Cat.No: T9710

Target: Cysteine Protease

Cat.No: T2493

Target: Cysteine Protease, Proteasome

Calpain Inhibitor XI

Cat.No: T72439

Calpain-2-IN-1

Cat.No: T63708

Neurodegenerative Disorder-Targeting Compound 1

Cat.No: T13486

Target: Others

Cat.No: T14187

Synonym: Calpain inhibitor II

Target: Others

Cat.No: T28786

Synonym: SJA-6017,Calpain Inhibitor VI,Calpain-In-4,SJA 6017,Calpain Inhibitor 4

Calpain inhibitor V

Cat.No: T80551

Synonym: Mu-Val-HPh-FMK

Target: Antibiotic

Z-Leu-Tyr-Chloromethylketone

Cat.No: T80103

Cat.No: T78632

Synonym: Calpain Inhibitor IV

Target: Proteasome

(Rac)-Neurodegenerative Disorder-Targeting Compound 1

Cat.No: T83527

Calpain Inhibitor XII

Cat.No: T21949

Acetyl-Calpastatin(184-210)(human) TFA

Cat.No: T75794

Ac-Leu-Leu-Norleucinol

Cat.No: T76364

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