Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6583 |
MG-101
ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I |
Cysteine Protease; Proteasome | Proteases/Proteasome; Ubiquitination |
MG-101 (Calpain inhibitor I) 是一种有效的半胱氨酸蛋白酶抑制剂,能够抑制钙蛋白酶I (Ki:190 pM),钙蛋白酶II (Ki:220 pM),组织蛋白酶B (Ki:150 pM)和组织蛋白酶L (Ki:500 pM)。 | |||
T6432 |
Calpeptin
|
Apoptosis; Cysteine Protease; Proteasome | Apoptosis; Proteases/Proteasome; Ubiquitination |
Calpeptin 是一种具有细胞穿透性的calpain 抑制剂,也是cathepsin K 抑制剂,其对人血小板 Calpain I 的ID50值为40 nM。 | |||
T21949 |
Calpain Inhibitor XII
|
||
(Rac)-Calpain Inhibitor XII是一种可逆的,选择性抑制钙蛋白酶I(calpain I; μ-calpain)的化合物,具有19 nM的Ki值。其对钙蛋白酶II(calpain II; m-calpain; Ki=120 nM)和组织蛋白酶B(cathepsin B; Ki=750 nM)显示出较低的抑制亲和力。(Rac)-Calpain Inhibitor XII用于研究钙蛋白酶在多种生理过程中的角色,如嗜中性粒细胞趋化性、神经元信号传导和心脏对损伤的响应。 | |||
TP2056 |
Acetyl-Calpastatin(184-210)(human)
Acetyl-Calpastatin (184-210) (human) |
||
Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio. |