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Cat. No. Product Name Target Signaling Pathways
T15038 Momelotinib sulfate

CYT387 sulfate salt

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Momelotinib sulfate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity versus JAK3.
T70823 Momelotinib HCl

Momelotinib HCl is a JAK1/2 inhibitor, reducing anemia in myelofibrosis (MF) patients.
T1849 Momelotinib

CYT11387,CYT387,LM-1149

Apoptosis; JAK; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Momelotinib (LM-1149) 是一种 ATP 竞争性的 JAK1/JAK2抑制剂,IC50值分别为 11 nM/18 nM。
T15037 Momelotinib Mesylate

CYT387 (Mesylate)

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Momelotinib Mesylate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity versus JAK3.

化合物

Momelotinib sulfate
Cat.No: T15038
Synonym: CYT387 sulfate salt
Target: JAK
Momelotinib HCl
Cat.No: T70823
Synonym:
Target:
Momelotinib
Cat.No: T1849
Synonym: CYT11387,CYT387,LM-1149
Target: Apoptosis, JAK, Autophagy
Momelotinib Mesylate
Cat.No: T15037
Synonym: CYT387 (Mesylate)
Target: JAK
TargetMol Loading
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