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Cat. No. Product Name Target Signaling Pathways
T2090 Lexibulin

CYT-997

Apoptosis; Reactive Oxygen Species; Microtubule Associated Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB
Lexibulin (CYT-997) 是一种微管蛋白聚集强效抑制剂,可诱导细胞凋亡,并诱导 GC 细胞中的线粒体ROS 生成。它对多种癌细胞的 IC50 值为 10-100n M,在体内外具有高细胞毒性和血管增生阻断作用。
T15746 Lexibulin dihydrochloride

CYT-997 dihydrochloride

Others Others
Lexibulin 2Hcl is an effective tubulin polymerization inhibitor (IC50: 10-100 nM in cancer cell lines). It also has potent cytotoxic and vascular disrupting activity in vitro and in vivo.

化合物

Lexibulin
Cat.No: T2090
Synonym: CYT-997
Target: Apoptosis, Reactive Oxygen Species, Microtubule Associated
Lexibulin dihydrochloride
Cat.No: T15746
Synonym: CYT-997 dihydrochloride
Target: Others
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