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Search Results for " ctr "

Targets Recommended: Somatostatin

31

抑制剂 & 化合物

2

天然产物

1

化合物库

7

重组蛋白

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Cat. No.	Product Name
L7860	Mini片段亲电杂环化合物库		369 compounds
	高溶解度共价杂环片段库中的 369 个化合物

化合物库

Mini片段亲电杂环化合物库

Cat.No: L7860

Compounds: 369

Cat. No.	Product Name	Target	Signaling Pathways
T2584	Octreotide SMS 201-995,奥曲肽	Somatostatin	GPCR/G Protein
	Octreotide (SMS 201-995) 是一种有效的生长激素、胰高血糖素和胰岛素抑制剂。它主要与生长抑素 2、3 和 5 亚型受体结合，可增强 Gi 活性，降低胞内 cAMP 的产生。
T4119	Octreotide Acetate 醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)	Somatostatin	GPCR/G Protein
	Octreotide Acetate (Sandostatin) 是一种长期有效的合成生长抑素八肽类似物，可抑制生长激素的分泌。
T67931	[Tyr3]Octreotate	Others	Others
	[Tyr3]Octreotate 是一个含有8个氨基酸的长肽化合物，是具有共价键DOTA 双功能螯合剂。[Tyr3]Octreotate 与SSR2活性的NETs 的跨膜受体结合，并通过内吞作用主动运输到细胞中，可能会增加所需的双链DNA 断裂，是治疗肿瘤的潜在药物。
T0340	Bisoctrizole Tinosorb M,UV-360,Milestab-360,紫外光吸收剂UV-360,Tinuvin-360	Others	Others
	Bisoctrizole (Tinosorb M) 是广谱紫外线吸收剂，能够吸收UVB 和UVA 射线，并反射和散射紫外线。
T68508	Ametoctradin
	Ametoctradin is a new Oomycete-specific fungicide and a potent Qo site inhibitor of the mitochondrial respiration complex III.
T76544	Cyclic SSTR agonist octreotide
	Cyclic SSTR agonist octreotide 是一种 Octreotide ，可作为生长抑素受体 (SSTR) 的激动剂。
T131601	Magnoflorine (Thalictrine; Esholine)
	Magnoflorine (Thalictrine; Esholine) 是一种有用的有机化合物，可用于生命科学领域的相关研究，其产品编号为 T131601。
T37300	PCTR1 PCTR1
	Protectin conjugates in tissue regeneration 1 (PCTR1) is a specialized pro-resolving mediator (SPM) synthesized from docosahexaenoic acid . DHA is oxidized to 16S,17S-epoxy-protectin, which is then converted to PCTR1 by glutathione S-transferase. PCTR1 levels increase during resolution of acute microbial-induced peritonitis in mice. PCTR1 (30 ng, i.p.) administration 12 hours post-infection increases macrophage numbers and activity and shortens the resolution phase of inflammation by 57%. It als...
T126238	Bionectriol A
	Bionectriol A 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T126238，CAS号为 1201896-30-1。
T37507	MCTR3 MCTR3
	Maresin conjugates in tissue regeneration 3 (MCTR3) is a specialized pro-resolving mediator (SPM) synthesized from docosahexaenoic acid in macrophages. DHA is oxidized to maresin 1 , which is converted to MCTR1 by glutathione S-transferase Mu 4 or leukotriene C4 synthase, then to MCTR2 by γ-glutamyl transferase, and to MCTR3 by dipeptidase. MCTR3 accelerates tissue regeneration in planaria (1 and 100 nM) approximately as potently as MCTR2 and more potently than MCTR1. Pretreatment with MCTR3 pri...
T37505	MCTR1 MCTR1
	Maresin conjugates in tissue regeneration 1 (MCTR1) is a specialized pro-resolving mediator (SPM) synthesized from docosahexaenoic acid in macrophages at the site of inflammation. DHA is oxidized to maresin 1 , which is then converted to MCTR1 by glutathione S-transferase Mu 4 or leukotriene C4 synthase. MCTR1 accelerates tissue regeneration in planaria (1 and 100 nM). Pretreatment with MCTR1 (50 ng/mouse, i.p.) prior to E. coli administration reduces neutrophil infiltration, shortens the inflam...
T37301	PCTR2
	Protein conjugates in tissue regeneration 2 (PCTR2) is a specialized pro-resolving mediator (SPM) synthesized from docosahexaenoic acid . DHA is oxidized to 16S,17S-epoxy-protectin, which is converted to PCTR1 by glutathione S-transferase and to PCTR2 via γ-glutamyl transpeptidase. PCTR2 is found in resolving mouse exudate and in both M1 and M2 macrophages differentiated from isolated human monocytes.
T80599	Dectrekumab QAX576
	Dectrekumab (QAX576) 是针对IL-13的人源化单克隆抗体。它能显著降低嗜酸性粒细胞性食管炎 (EoE) 患者上皮内的嗜酸性粒细胞数量，并改善食管疾病相关的转录失调情况，适用于免疫炎症研究。
T38443	Methoctramine tetrahydrochloride
	Methoctramine tetrahydrochloride is a potent and cardioselective antagonist of the M2 muscarinic receptor, capable of inhibiting Muscarine-induced bradycardia in vivo.
T37728	Methoctramine (hydrate)
	Methoctramine is a selective antagonist of M2 muscarinic acetylcholine receptors (IC50 = 6.1 nM in CHO-K1 cell membranes).[1] It is selective for M2 over M1, M3, M4, and M5 receptors (IC50s = 92, 770, 260, and 217 nM, respectively). In vitro, methoctramine inhibits acetylcholine-induced reductions in isolated guinea pig tracheal tube contractions when used at a concentration of 1 μM.[2] In vivo, methoctramine inhibits bradycardia and bronchoconstriction induced by acetylcholinein guinea pigs wit...
T37302	PCTR3
	Protein conjugates in tissue regeneration 3 (PCTR3) is a specialized pro-resolving mediator (SPM) synthesized from docosahexaenoic acid . DHA is oxidized to 16S,17S-epoxy-protectin, which is converted to PCTR1 by glutathione S-transferase and to PCTR2 and PCTR3 via peptidases. PCTR3 is found in infected mouse spleens and resolving exudate as well as isolated human spleen and septic plasma. It is also found in both M1 and M2 macrophages differentiated from isolated human monocytes.
T2584L2	Octreotide pamoate SMS pa,SMS 201-995 pa
	Octreotide pamoate is an antineoplastic agent.
T37506	MCTR2 MCTR2
	Maresin conjugates in tissue regeneration 2 (MCTR2) is a specialized pro-resolving mediator (SPM) synthesized from docosahexaenoic acid in macrophages at the site of inflammation. DHA is oxidized to maresin 1 , which is converted to MCTR1 by glutathione S-transferase Mu 4 or leukotriene C4 synthase then to MCTR2 by γ-glutamyl transferase. MCTR2 accelerates tissue regeneration in planaria (1 and 100 nM). Pretreatment with MCTR2 prior to E. coli administration reduces neutrophil infiltration, shor...
T71130	Spectramide
	Spectramide is a dopamine D-2 receptor antagonist.
T71557	3-Tyr-octreotide
	3-Tyr-octreotide is a biochemical that has been evaluated for tumor inhibition.
T83191	Acetyl-Lys5-octreotide
	Acetyl-Lys5-octreotide为一生物活性肽，具备特定的生理和生化作用。
T19240	Cinoctramide	Others	Others
	Cinoctramide is a pharmaceutical intermediate.
T68628	Plectranthoic Acid
	Plectranthoic Acid is an activator of AMPK which induces apoptotic death in prostate cancer cells.
T124624	Nectriapyrone
	Nectriapyrone 是一种有用的有机化合物，可用于生命科学领域的相关研究。其产品编号为 T124624，CAS号为 57685-79-7。
T2584L1	Octreotide HCl Octreotide hydrochloride, (-)-,Octreotide hydrochloride
	Octreotide HCl is a potent, long-acting synthetic SOMATOSTATIN octapeptide analog that inhibits the secretion of growth hormone.
T37166	RCTR1
	Resolvin conjugate in tissue regeneration 1 (RCTR1) is a specialized pro-resolving mediator (SPM) biosynthesized from docosahexaenoic acid by isolated human macrophages and apoptotic polymorphonuclear (PMN) neutrophils.1It has been found in human spleen and bone marrow.2RCTR1 is produced via lipoxygenase-mediated oxidation of DHA to 7(S)-8-epoxy-17(S)-HDHA, which is conjugated to glutathione.1,2,3RCTR1 (10 nM) increases phagocytosis ofE. colior apoptotic neutrophils in isolated human monocyte-de...
T6590	MK-3207 Hydrochloride MK-3207 HCl	CGRP Receptor	GPCR/G Protein; Neuroscience
	MK-3207 Hydrochloride (MK-3207 HCl) 是口服具有活力的CGRP receptor 拮抗剂，IC50=0.12 nM，Ki=0.024 nM。
T76262L	Cagrilintide acetate
	Cagrilintide acetate 是一种非选择性的 AMYR/CTR 激动剂和长效酰化淀粉酶类似物。Cagrilintide acetate 以剂量依赖的方式导致食物摄入减少和体重明显下降。Cagrilintide acetate 可用于肥胖症的研究。
T76262	Cagrilintide
	Cagrilintide为一种处于研发阶段的新型长效酰化胰岛素类似物，兼具非选择性胰岛素受体(AMYR)与降钙素G蛋白偶联受体(CTR)的激动剂功能。该化合物能显著降低体重并减少食物摄入，展现出针对肥胖疾病的研究潜力。
T37413	Calcitonin (salmon) (trifluoroacetate salt)
	Calcitonin is a peptide hormone that lowers blood calcium level and inhibits bone resorption. It belongs to the calcitonin family of peptides, which also includes amylin , calcitonin gene-related peptide , and adrenomedullin. The binding of salmon calcitonin to the human calcitonin receptor (CTR) is not modulated by receptor activity-modifying proteins (RAMPs), which influence affinity of human calcitonin to CTR. Salmon calcitonin binds to human CTR2 with IC50 values of 0.933, 0.224, 0.134, and ...
T21558	MK-3207
	MK-3207是口服生物相容性的CGRP 受体拮抗剂，IC50和 Ki 分别为 0.12 nM 和 0.024 nM，对 AM1，AM2，CTR 和 AMY3 的抑制性较弱。MK-3207可用于偏头痛研究。

化合物

Cat.No: T2584

Synonym: SMS 201-995,奥曲肽

Target: Somatostatin

Octreotide Acetate

Cat.No: T4119

Synonym: 醋酸奥曲肽,SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)

Target: Somatostatin

[Tyr3]Octreotate

Cat.No: T67931

Target: Others

Cat.No: T0340

Synonym: Tinosorb M,UV-360,Milestab-360,紫外光吸收剂UV-360,Tinuvin-360

Target: Others

Cat.No: T68508

Cyclic SSTR agonist octreotide

Cat.No: T76544

Magnoflorine (Thalictrine; Esholine)

Cat.No: T131601

Cat.No: T37300

Synonym: PCTR1

Cat.No: T126238

Cat.No: T37507

Synonym: MCTR3

Cat.No: T37505

Synonym: MCTR1

Cat.No: T37301

Cat.No: T80599

Synonym: QAX576

Methoctramine tetrahydrochloride

Cat.No: T38443

Methoctramine (hydrate)

Cat.No: T37728

Cat.No: T37302

Octreotide pamoate

Cat.No: T2584L2

Synonym: SMS pa,SMS 201-995 pa

Cat.No: T37506

Synonym: MCTR2

Cat.No: T71130

3-Tyr-octreotide

Cat.No: T71557

Acetyl-Lys5-octreotide

Cat.No: T83191

Cat.No: T19240

Target: Others

Plectranthoic Acid

Cat.No: T68628

Cat.No: T124624

Cat.No: T2584L1

Synonym: Octreotide hydrochloride, (-)-,Octreotide hydrochloride

Cat.No: T37166

MK-3207 Hydrochloride

Cat.No: T6590

Synonym: MK-3207 HCl

Target: CGRP Receptor

Cagrilintide acetate

Cat.No: T76262L

Cat.No: T76262

Calcitonin (salmon) (trifluoroacetate salt)

Cat.No: T37413

Cat.No: T21558

Cat. No.	Product Name	Target	Signaling Pathways
TN1139L	Tetradehydrothalictrifoline	Others	Others
	Tetradehydrothalictrifoline 是一种天然产品。
T1683	Actriol 异雌三醇,Epiestriol	Glucocorticoid Receptor	Endocrinology/Hormones
	Actriol (Epiestriol) 是内源性雌激素雌酮的代谢物，拥有抗炎及抗菌活性。

天然产物

Tetradehydrothalictrifoline

Cat.No: TN1139L

Target: Others

Cat.No: T1683

Synonym: 异雌三醇,Epiestriol

Target: Glucocorticoid Receptor

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPY-00317	Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc) CTR,calcitonin receptor,CRT,CTR1,CT-R	Human	HEK293 Cells
	Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 43.9 kDa and the accession number is P30988-1.
TMPY-00085	Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc) CTR,CTR1,CT-R,calcitonin receptor,CRT	Human	HEK293 Cells
	Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.1 kDa and the accession number is P30988-2.
TMPY-00215	CTRB1 Protein, Rat, Recombinant (His) chymotrypsinogen B1	Rat	HEK293 Cells
	CTRB1 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.4 kDa.
TMPH-02595	Collectrin Protein, Mouse, Recombinant (His & Myc & SUMO) Cltrn,Collectrin,Tmem27,Nx17,Transmembrane protein ...	Mouse	E. coli
	Plays an important role in amino acid transport by acting as binding partner of amino acid transporters SLC6A18 and SLC6A19, regulating their trafficking on the cell surface and their activity. May also play a role in trafficking of amino acid transporters SLC3A1 and SLC7A9 to the renal cortical cell membrane. Regulator of SNARE complex function. Stimulator of beta cell replication.
TMPY-03653	CTRL Protein, Human, Recombinant (His) CTRL1,chymotrypsin-like	Human	HEK293 Cells
	CTRL-1, also known as chymotrypsin-like protease, belongs to thepeptidase S1 family. CTRL-1 contains 1peptidase S1 domain. Its expression is increased in preeclampsia (PE). Placental-derived chymotrypsin-like protease is responsible for inducing endothelial inflammatory phenotypic changes possibly by upregulation of cell adhesion molecule expressions, activation of cellular protease, and induction of extracellular regulated kinase phosphorylation. Activated microglia have been observed in variou...
TMPJ-00881	CTRB1 Protein, Human, Recombinant (His) CTRB,CTRB1,Chymotrypsinogen B	Human	HEK293 Cells
	Chymotrypsinogen B (CTRB1) is a 263 amino acid protein with signal peptide (1-18) and Chymotrypsinogen B (19-263). Chymotrypsinogen B have three chains:Chymotrypsin B chain A(19-31), Chymotrypsin B chain B(34-164), Chymotrypsin B chain C (167-263). Chymotrypsinogen B is a Serine Protease Hydrolase secrets into gastrointestinal tract as the inactive precursor Chymotrypsinogen.
TMPY-00358	Arp3/ACTR3 Protein, Human, Recombinant (His & GST) ARP3,ARP3 actin-related protein 3 homolog (yeast)	Human	Baculovirus Insect Cells
	Arp3/ACTR3 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 75.1 kDa and the accession number is A0A024RAI1.

重组蛋白

Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc)

Cat.No: TMPY-00317

Species: Human

Expression System: HEK293 Cells

Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc)

Cat.No: TMPY-00085

Species: Human

Expression System: HEK293 Cells

CTRB1 Protein, Rat, Recombinant (His)

Cat.No: TMPY-00215

Species: Rat

Expression System: HEK293 Cells

Collectrin Protein, Mouse, Recombinant (His & Myc & SUMO)

Cat.No: TMPH-02595

Species: Mouse

Expression System: E. coli

CTRL Protein, Human, Recombinant (His)

Cat.No: TMPY-03653

Species: Human

Expression System: HEK293 Cells

CTRB1 Protein, Human, Recombinant (His)

Cat.No: TMPJ-00881

Species: Human

Expression System: HEK293 Cells

Arp3/ACTR3 Protein, Human, Recombinant (His & GST)

Cat.No: TMPY-00358

Species: Human

Expression System: Baculovirus Insect Cells

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