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Cat. No. Product Name Target Signaling Pathways
T2262 Itanapraced

CHF5074,CSP-1103

Beta Amyloid; Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
Itanapraced (CHF5074) 是新型γ-secretase 调节剂,能够降低 Aβ42 (IC50=3.6 nM) 和 Aβ40 (IC50=18.4 nM) 分泌。
T69061 CSP-2503

CSP-2503 is a 5-HT1A receptor agonist.
T38559 Competence-Stimulating Peptide-2 (CSP-2)

Competence-Stimulating Peptide-2 (CSP-2) is a quorum sensing signal peptide synthesized by Streptococcus pneumoniae. ComD2, a compatible receptor of CSP-2, exhibits an EC 50 value of 50.7 nM.
T39175 CSP1

CSP1 is a highly potent and selective agonist of the ComD1 receptor, exhibiting an IC50 value of 10.3 nM. It represents a major variant of competence-stimulating peptide (CSP) and plays a crucial role in regulating the genetic transformation of S. pneumoniae through modulation of quorum sensing (QS). Additionally, CSP1 possesses antibacterial activity, further enhancing its potential as an effective antibacterial agent.
T8778 TTK21

Epigenetic Reader Domain Chromatin/Epigenetic
TTK21 是 CBP/p300 组蛋白乙酰转移酶活性的激活剂,与葡萄糖基碳纳米球结合时,可通过血脑屏障,对成人大脑神经发生和长期记忆功能有益。
T63163 cSPM

cSPM (Cyclic spermine) 是一种 Aβ42 抑制剂。cSPM 对三种不同肽 Aβ42、胰淀素和胰岛素的聚集具有抑制作用,且能够减少细胞毒性。
T21220 3-Chlorodiphenylamine

3-Cl DPA,3-氯二苯胺,3-Cl-DPA,3 Cl-DPA

3-Cl-DPA, a cardiac troponin activator, acts by a mechanism distinct from bepridil or TFP.

化合物

Itanapraced
Cat.No: T2262
Synonym: CHF5074,CSP-1103
Target: Beta Amyloid, Gamma-secretase
CSP-2503
Cat.No: T69061
Synonym:
Target:
Competence-Stimulating Peptide-2 (CSP-2)
Cat.No: T38559
Synonym:
Target:
CSP1
Cat.No: T39175
Synonym:
Target:
TTK21
Cat.No: T8778
Synonym:
Target: Epigenetic Reader Domain
cSPM
Cat.No: T63163
Synonym:
Target:
3-Chlorodiphenylamine
Cat.No: T21220
Synonym: 3-Cl DPA,3-氯二苯胺,3-Cl-DPA,3 Cl-DPA
Target:
TargetMol Loading
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