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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T69981 |
CRM-51005
|
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CRM-51005 is a new phospholipase C inhibitor produced by unidentified fungal strain MT51005 | |||
T69980 |
XMU-MP-2
|
BTK; Protease | Angiogenesis; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
XMU-MP-2 是一种有效和选择性的蛋白酶抑制剂,具有抗癌活性,在小鼠异种移植模型中 抑制致癌 BRK 驱动的肿瘤的生长。 | |||
T26624 |
AN0128
AN 0128,CRM-0005,CRM0005,ONT0001,AN-0128,ONT-0001 |
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AN 0128 is a tumour necrosis factor alpha (TNF-α) inhibitor. | |||
T79654 |
CRM1-IN-1
|
CRM1 | Membrane transporter/Ion channel |
CRM1-IN-1 (Compound KL1) 为非共价CRM1抑制剂,能诱导核CRM1降解(IC50: 0.27 μM),抑制CRM1介导的核输出与细胞增殖,同时触发结直肠癌细胞凋亡 (apoptosis)。 | |||
T79655 |
CRM1-IN-2
|
CRM1 | Membrane transporter/Ion channel |
CRM1-IN-2(Compound KL2)为非共价CRM1抑制剂,能够定位CRM1于核外围,耗尽核内CRM1,从而抑制CRM1介导的核输出。该化合物能抑制结直肠癌细胞的生长并诱导细胞凋亡(apoptosis)。 | |||
T60416 | CRM1 degrader 1 | ||
CRM1 degrader 1 (1l) 是一种低毒的CRM1降解剂,可诱导胃癌细胞凋亡并选择性抑制胃癌细胞的增殖。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN5131 |
Tetrahydrocannabivarin
THCV,delta9-Tetrahydrocannabivarin,CRM,Tetrahydrocannavarin |
Cannabinoid Receptor | GPCR/G Protein |
Tetrahydrocannabivarin (CRM) 是 cannabinoid type 1 receptor 的中性拮抗剂,对 2 型糖尿病有潜在治疗价值。 |