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Cat. No. Product Name Target Signaling Pathways
T0373L Erlotinib hydrochloride

盐酸埃罗替尼,OSI-744,NSC 718781,Erlotinib HCl,CP-358774

EGFR; Autophagy Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Erlotinib hydrochloride (NSC 718781) 抑制EGFR 激酶的IC50为 2 nM,用于治疗非小细胞肺癌。
T0373 Erlotinib

OSI-744,NSC 718781,CP358774,埃罗替尼,R1415

EGFR; Autophagy Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Erlotinib (NSC-718781) 是一种直接作用的EGFR 酪氨酸激酶抑制剂,用于治疗非小细胞肺癌,对人 EGFR 的IC50为 2 nM。它可降低完整肿瘤细胞的 EGFR 自磷酸化,IC50为 20 nM。
T0373L1 Erlotinib mesylate

CP-358774,CP-358,774,埃罗替尼甲磺酸盐,OSI-774,CP358774,OSI 774

Erlotinib is an epidermal growth factor receptor inhibitor. Erlotinib binds in a reversible fashion to the adenosine triphosphate (ATP) binding site of the receptor.
T11229 Erlotinib-d6

OSI-774 D6,NSC 718781 D6,CP-358774 D6

Others Others
Erlotinib is a directly acting inhibitor EGFR tyrosine kinase inhibitor with an IC50 of 2 nM for human EGFR. Erlotinib D6 is a deuterium labeled Erlotinib .
T19312 Erlotinib-d6 hydrochloride

CP-358774 D6 hydrochloride,NSC 718781 D6 hydrochloride,Erlotinib D6 hydrochloride,OSI-774 D6 hydrochloride

Others Others
Erlotinib Hydrochloride inhibits purified EGFR kinase with an IC50 of 2 nM. Erlotinib D6 hydrochloride a deuterium labeled Erlotinib Hydrochloride.
T35915 Erlotinib-13C6

Erlotinib-13C6

Erlotinib-13C6 (CP-358774-13C6) is a 13C-labeled Erlotinib. Erlotinib is a directly acting EGFR tyrosine kinase inhibitor, with an IC50 of 2 nM for human EGFR[1]. Erlotinib reduces EGFR autophosphorylation in intact tumor cells with an IC50 of 20 nM. Erlotinib is used for the treatment of non-small cell lung cancer[1].Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process[2]...

化合物

Erlotinib hydrochloride
Cat.No: T0373L
Synonym: 盐酸埃罗替尼,OSI-744,NSC 718781,Erlotinib HCl,CP-358774
Target: EGFR, Autophagy
Erlotinib
Cat.No: T0373
Synonym: OSI-744,NSC 718781,CP358774,埃罗替尼,R1415
Target: EGFR, Autophagy
Erlotinib mesylate
Cat.No: T0373L1
Synonym: CP-358774,CP-358,774,埃罗替尼甲磺酸盐,OSI-774,CP358774,OSI 774
Target:
Erlotinib-d6
Cat.No: T11229
Synonym: OSI-774 D6,NSC 718781 D6,CP-358774 D6
Target: Others
Erlotinib-d6 hydrochloride
Cat.No: T19312
Synonym: CP-358774 D6 hydrochloride,NSC 718781 D6 hydrochloride,Erlotinib D6 hydrochloride,OSI-774 D6 hydrochloride
Target: Others
Erlotinib-13C6
Cat.No: T35915
Synonym: Erlotinib-13C6
Target:
TargetMol Loading
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