Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T10840 |
CM-579 trihydrochloride (1846570-40-8 free base)
CM-579 trihydrochloride |
DNA Methyltransferase | Chromatin/Epigenetic |
CM-579 trihydrochloride is a first-in-class reversible and dual inhibitor of G9a and DNMT (IC50s: 16 nM, 32 nM) with potent in vitro cellular activity in a wide range of cancer cells. | |||
T72277 |
CM-579 trihydrochloride
|
||
CM-579 trihydrochloride 是首创的、可逆的,G9a 和 DNA 甲基转移酶(DNMT)的双抑制剂,其 IC50值分别为 16 nM 和32 nM。在多种癌细胞中发挥有效活性作用。 | |||
T10840L |
CM-579
|
DNA Methyltransferase; Histone Methyltransferase | Chromatin/Epigenetic |
CM-579 是首创的、可逆的,G9a 和 DNA 甲基转移酶 (DNMT) 的双抑制剂,其 IC50 值分别为 16 nM 和32 nM。在多种癌细胞中发挥有效活性作用。 |