Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T17305 |
CDK8-IN-4
|
CDK | Cell Cycle/Checkpoint |
CDK8-IN-4 is an inhibitor of CDK8 (IC50: 0.2 nM). | |||
T72048 |
CDK8-IN-12
|
GSK-3; CDK | Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells |
CDK8-IN-12 是一种具有选择性、有效性和口服活性的 CDK8 抑制剂(Ki : 14 nM),是一种抗癌剂。CDK8-IN-12 对 GSK-3α、GSK-3β、PCK-θ 具有抑制作用,Ki 分别为 13 nM、4 nM、109 nM。CDK8-IN-12对 MV4-11 细胞显示出抗增殖活性。 |