Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T20324 |
Butyrophenone
苯丁酮,NSC8463,NSC 8463,NSC-8463 |
Others | Others |
Butyrophenone (NSC-8463) 是一种化合物。它的一些衍生物用于治疗各种精神疾病。 | |||
T7421 |
Melperone
|
Others | Others |
Melperone 是一种丁酰苯,是一种具有睡眠诱导作用的抗精神病试剂,常用于研究精神类疾病。 | |||
T6398 |
Azaperone
R-1929,Fluoperidol,阿扎哌隆,Stresnil,NSC 170976,Suicalm |
Others; Dopamine Receptor | GPCR/G Protein; Neuroscience; Others |
Azaperone (Fluoperidol) 是多巴胺拮抗剂,具有一些抗组胺和抗胆碱特性,具有止吐活性。 | |||
T14830 |
Bromperidol
溴哌利多,R-11333 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Bromperidol (R-11333) 是一种苯丁酮衍生物,是一种强效长效精神安定药。它被用作治疗精神分裂症的抗精神病药。 | |||
T4275 |
Fluanisone
Sedalande,氟苯丙酮哌嗪,Haloanison |
Others | Others |
Fluanisone (Haloanison) 是一种苯丁酮衍生物,具有镇静作用。它是一种典型的抗精神病药,用于治疗精神分裂症。 | |||
T0280 |
Spiperone
螺哌隆,Spiroperidol,Spiropitan |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Spiperone (Spiropitan) 是多巴胺 D2、血清素5-HT1A 和血清素5-HT2A 拮抗剂。它是广泛使用的药理学工具。它具有研究神经系统疾病的潜力。 | |||
T25661 |
Lenperone
Lenperonum,AHR-2277 [as hydrochloride] |
||
Lenperone is a butyrophenone antipsychotic. Like other major tranquilizers, It has some alpha-adrenergic blocking action and is antiemetic. | |||
T29750 |
AHR-1900 hydrochloride
AHR-1900 HCl |
||
AHR-1900 hydrochloride is a butyrophenone derivative used in the treatment of schizophrenia. | |||
T29750L |
AHR-1900 free base
AHR-1900, |
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AHR-1900 free base is a butyrophenone derivative which may be used in the treatment of schizophrenia. | |||
T71926 |
Melperone hydrochloride
|
||
Melperone hydrochloride is a butyrophenone neuroleptic and an inhibitor of the CYP2D6 catalyzed O-demethylation of venlafaxine. |