Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5850 |
Benzamil
Benzamil (hydrochloride) |
Na+/Ca2+ Exchanger; Sodium Channel | Membrane transporter/Ion channel |
Benzamil 是 Amiloride 类似物,是 Na+/Ca2+交换体抑制剂,抑制 TRPP3 介导的 Ca2+激活电流,IC50为 1.1 μM。它也是一种非选择性上皮钠通道 (ENaC) 阻滞剂,能增强肌源性血管收缩。 | |||
T22266 |
Benzamil hydrochloride
Benzylamiloride hydrochloride,3,5-二氨基-N-[(E)-氨基(苄基氨基)亚甲基]-6-氯-2-吡嗪甲酰胺盐酸盐(1:1) |
Others | Others |
Benzamil hydrochloride is a specific and potent sodium channel (ENaC) blocker. | |||
T26383 |
3',4'-Dichlorobenzamil HCl
|
||
3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels. |