Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T70875 |
BI-665915
|
||
BI-665915 is a 5-lipoxygenase activating protein inhibitor. | |||
T70873 |
M3541
|
Apoptosis; ATM/ATR | Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
M3541 是一种具有选择性有效性和口服活性的 ATM 抑制剂,具有潜在抗肿瘤活性。M-3541 通过与 ATM 结合来抑制 ATM 的激酶活性和 ATM 介导的信号传导。M3541 防止 DNA 损伤检查点激活,抑制 DNA 损伤修复,促使肿瘤细胞凋亡,并诱导 ATM 过表达的肿瘤细胞死亡。 | |||
T12793 |
(S)-BI 665915
|
Others | Others |
(S)-BI 665915 is an orally active inhibitor of oxadiazole-containing 5-lipoxygenase-activating protein (FLAP)(IC50 of 1.7 nM for FLAP binding).. |