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Cat. No. Product Name Target Signaling Pathways
T34925 Triafamone

BCS BX60309,BCSBX60309,BCS-BX60309

Triafamone is a new sulfonanilide herbicide.
T13176 TNO155

Batoprotafib

Phosphatase Metabolism
TNO155 是具有口服活性野生型SHP2的选择性变构抑制剂 (IC50= 0.011 µM)。它有研究 RTK 依赖性恶性肿瘤(尤其是晚期实体瘤)的潜力。
T7679 UBCS039

Sirtuin; Autophagy Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair
UBCS039 是一种合成的 SIRT6特异性激活剂,可在人癌细胞中诱导自噬,其 EC50值为38 μM。
T70908 EST64454 free base

EST64454 is a σ1 receptor (σ1R) antagonist clinical candidate for the treatment of pain. EST64454 shows an outstanding aqueous solubility, which together with its high permeability in Caco-2 cells will allow its classification as a BCS class I compound. It also shows high metabolic stability.

化合物

Triafamone
Cat.No: T34925
Synonym: BCS BX60309,BCSBX60309,BCS-BX60309
Target:
TNO155
Cat.No: T13176
Synonym: Batoprotafib
Target: Phosphatase
UBCS039
Cat.No: T7679
Synonym:
Target: Sirtuin, Autophagy
EST64454 free base
Cat.No: T70908
Synonym:
Target:
TargetMol Loading
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