Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T14998 |
Copanlisib dihydrochloride
库潘尼西盐酸,BAY 80-6946 dihydrochloride |
Apoptosis; PI3K; mTOR | Apoptosis; PI3K/Akt/mTOR signaling |
Copanlisib dihydrochloride (BAY 80-6946 dihydrochloride) 是一种选择性和 ATP 竞争性的泛 I 类 PI3K 抑制剂。它具有优越的抗肿瘤活性,对除 mTOR 以外的其他脂质和蛋白激酶的选择性也超过 2,000 倍。 | |||
T6322 |
Copanlisib
BAY 80-6946,可泮利塞,库潘尼西 |
Apoptosis; PI3K | Apoptosis; PI3K/Akt/mTOR signaling |
Copanlisib (BAY 80-6946) 是一种选择性的和 ATP 竞争性的泛 I 类PI3K 抑制剂,具有抗肿瘤活性,对PI3Kα,PI3Kδ,PI3Kβ和PI3Kγ的IC50分别为 0.5 nM、0.7 nM、3.7 nM 和 6.4 nM。 | |||
T70756 |
KT172
|
||
KT172 是一种 DAGLβ抑制剂,IC50值为 11 nM。KT172 可用于代谢和炎症的研究。 | |||
T35534 |
7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine
|
||
7-Methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-amine is a building block.1It has been used in the synthesis of PI3K inhibitors. 1.Scott, W.J., Hentemann, M.F., Rowley, R.B., et al.Discovery and SAR of novel 2,3-dihydroimidazo[1,2-c]quinazoline PI3K inhibitors: Identification of copanlisib (BAY 80-6946)ChemMedChem.11(14)1517-1530(2016) |