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Search Results for " bace1-in-5 "

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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T10453 BACE1-IN-5

Beta Amyloid; BACE Neuroscience
BACE1-IN-5 (Compound 15) 是一种 BACE1抑制剂,IC50为 9.1 nM。BACE1-IN-5还可抑制细胞 Aβ,IC50为 0.82 nM。并且,BACE1-IN-5 具有改善 hERG 抑制和 P-gp 外排的药物化学作用。
T35975 6,9-Dichloro-1,2,3,4-tetrahydroacridine

6,9-Dichloro-1,2,3,4-tetrahydroacridine is a synthetic intermediate in the synthesis of tacrine-based acetylcholinesterase (AChE) inhibitors.1It is also an intermediate in the synthesis of multifunctional tacrine hybrids that possess radical scavenging, amyloid-β aggregation inhibitory, and/or β-secretase 1 (BACE1) inhibitory activities in addition to their activity as AChE inhibitors.2,3 1.Recanatini, M., Cavalli, A., Belluti, F., et al.SAR of 9-amino-1,2,3,4-tetrahydroacridine-based acetylchol...

化合物

BACE1-IN-5
Cat.No: T10453
Synonym:
Target: Beta Amyloid, BACE
6,9-Dichloro-1,2,3,4-tetrahydroacridine
Cat.No: T35975
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4115 Auraptene

橙皮油内酯,7-geranyloxycoumarin,橙皮油素

MMP; BACE Neuroscience; Proteases/Proteasome
Auraptene 是一种丰富的天然香叶氧基香豆素。它能够抑制基质金属蛋白酶 2 以及关键炎症因子,包括 IL-6,IL-8 和趋化因子 (C-C 基序) 配体-5 (CCL5)的分泌。

天然产物

Auraptene
Cat.No: T4115
Synonym: 橙皮油内酯,7-geranyloxycoumarin,橙皮油素
Target: MMP, BACE
TargetMol Loading
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